SCHEMBL8201557

SCHEMBL8201557

CNc1ncnc(OC)c1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.49
PDPK1 O15530 2/20 0.40
YTHDC1 Q96MU7 2/20 0.39
YTHDF2 Q9Y5A9 1/20 0.39
ALDH1A1 P00352 4/20 0.37
HSD17B10 Q99714 4/20 0.37
CYP1A2 P05177 4/20 0.37
CYP3A4 P08684 3/20 0.37
TDP1 Q9NUW8 2/20 0.37
LCK P06239 4/20 0.36
LMNA P02545 3/20 0.36
CYP2C19 P33261 3/20 0.36
CYP2D6 P10635 2/20 0.36
USP2 O75604 1/20 0.36
CYP2C9 P11712 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
EGFR P00533 3/20 0.35
GAK O14976 2/20 0.35
SRC P12931 1/20 0.35
KDM4E B2RXH2 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3817132 0.79 PDPK1 (0.45) ESR1PDPK1ALDH1A1HSD17B10CYP1A2
SCHEMBL12261899 0.79 YTHDC1 (0.39) ESR1PDPK1YTHDC1YTHDF2ALDH1A1
SCHEMBL9046753 0.78 PGK1 (0.41) PDPK1YTHDC1YTHDF2ALDH1A1HSD17B10
SCHEMBL24344244 0.78 ALDH1A1 (0.36) ESR1PDPK1YTHDC1YTHDF2ALDH1A1
SCHEMBL9050477 0.74 ESR1 (0.46) ESR1ALDH1A1CYP1A2LMNACYP2D6
SCHEMBL23326914 0.73 ESR1 (0.38) ESR1PDPK1YTHDC1YTHDF2ALDH1A1
SCHEMBL14326156 0.71 PDPK1 (0.39) ESR1PDPK1ALDH1A1HSD17B10CYP1A2
SCHEMBL11771336 0.70 PDPK1 (0.38) ESR1PDPK1ALDH1A1LCKHPGD
SCHEMBL9044468 0.70 ALDH1A1 (0.39) ESR1PDPK1ALDH1A1TDP1LCK
SCHEMBL6233405 0.70 PDE5A (0.46) ESR1PDPK1LCKLMNAEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008097546-A2 COMPOUNDS THAT INHIBIT CHOLINESTERASE COLUCID PHARMACEUTICALS, INC. (US) 2008-08-14 WO disclosed