SCHEMBL9051204

SCHEMBL9051204

CCCc1cc(CBr)ccc1OOC(=O)Cc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
TSHR P16473 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPK1 P28482 1/20 0.36
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
PAM P19021 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9058139 0.89 CYP1A2 (0.39) CYP1A2CYP3A4CYP2C19TSHRL3MBTL1
SCHEMBL9447429 0.78 CHRM1 (0.52) L3MBTL1
SCHEMBL9051202 0.73 EDNRB (0.55)
SCHEMBL7410289 0.71 PPARG (0.50) ALDH1A1
SCHEMBL9126741 0.68 PPARG (0.47) ALDH1A1
SCHEMBL14420218 0.68 TLR7 (0.51) TSHRALDH1A1
SCHEMBL9165064 0.68 PPARD (0.42) TSHRALDH1A1MAPK1
SCHEMBL2817717 0.67 CYP3A4 (0.56) CYP1A2CYP3A4CYP2C19L3MBTL1ALDH1A1
SCHEMBL664857 0.66 ALDH1A1 (0.65) TSHRL3MBTL1ALDH1A1MAPK1PAM
Benzene SCHEMBL9407299 0.66 ALDH1A1 (0.65) TSHRL3MBTL1ALDH1A1MAPK1PAM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0515535-A4 ANGIOTENSIN II ANTAGONISTS INCORPORATING A SUBSTITUTED BENZYL ELEMENT MERCK & CO INC (US) 1996-01-17 EP disclosed
US-5420133-A Quinazolinones substituted with phenoxyphenylacetic acid derivatives MERCK & CO., INC. (US) 1995-05-30 US disclosed
US-5401745-A Cardiovascular disorders or hypotensive agents MERCK & CO., INC. (US) 1995-03-28 US disclosed
WO-1994021259-A1 QUINAZOLINONES SUBSTITUTED WITH PHENOXYPHENYLACETIC ACID DERIVATIVES MERCK & CO., INC. (US) 1994-09-29 WO disclosed
US-5264439-A Quinazolinone, triazolinone and pyrimidinone angiotensin II antagonists incorporating a substituted benzyl element MERCK & CO., INC. (US) 1993-11-23 US disclosed
EP-0515535-A1 ANGIOTENSIN II ANTAGONISTS INCORPORATING A SUBSTITUTED BENZYL ELEMENT MERCK & CO. INC. (US) 1992-12-02 EP disclosed
WO-1991012001-A1 ANGIOTENSIN II ANTAGONISTS INCORPORATING A SUBSTITUTED BENZYL ELEMENT MERCK & CO., INC. (US) 1991-08-22 WO disclosed