SCHEMBL9051254

SCHEMBL9051254

O=C(O)c1cccc(Oc2cccc(CN(Cc3ccc([N+](=O)[O-])cc3)C(c3c[nH]cn3)C(c3ccccc3)(c3ccccc3)c3ccccc3)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
FFAR1 O14842 2/20 0.41
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
SLC2A1 P11166 1/20 0.38
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CETP P11597 1/20 0.36
FAAH O00519 1/20 0.36
MGLL Q99685 1/20 0.36
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36
MMP13 P45452 1/20 0.36
LPAR1 Q92633 2/20 0.35
LPAR5 Q9H1C0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9056541 0.93 FFAR1 (0.41) KDM4EFFAR1MEN1KMT2ASLC2A1
SCHEMBL9052107 0.81 NR3C1 (0.39) KDM4EFFAR1ALDH1A1LMNASMN1; SMN2
SCHEMBL9050102 0.78 NR3C1 (0.45) KDM4EFFAR1MEN1KMT2AALDH1A1
SCHEMBL177838 0.67 KDM4E (1.00) KDM4EFFAR1MEN1KMT2AALDH1A1
SCHEMBL8644568 0.66 AKR1C3 (0.39)
SCHEMBL7044513 0.65 MAOB (0.79) KDM4EMEN1KMT2AMAOAMAOB
Hydrochloric Acid SCHEMBL8351982 0.63 KMT2A (0.39) MEN1KMT2ALMNASMN1; SMN2
SCHEMBL9054914 0.61 AKR1C3 (0.44) KDM4E
SCHEMBL13240466 0.60 TP53 (0.61) KDM4EMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL11265703 0.60 MAOB (0.79) MAOAMAOBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996037204-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1996-11-28 WO disclosed