SCHEMBL9051259

SCHEMBL9051259

CS(=O)(=O)N(c1ccccc1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.47
TACR1 P25103 5/20 0.46
CTSD P07339 6/20 0.40
BACE1 P56817 6/20 0.40
BACE2 Q9Y5Z0 6/20 0.40
NR1H3 Q13133 1/20 0.40
MAPT P10636 1/20 0.39
HSD11B1 P28845 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
RORC P51449 2/20 0.37
P2RX1 P51575 1/20 0.37
ACP1 P24666 1/20 0.37
PTPN7 P35236 1/20 0.37
PTPN12 Q05209 1/20 0.37
PTPN13 Q12923 1/20 0.37
SSU72 Q9NP77 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8659812 0.82 PKM (0.54) L3MBTL1TACR1NR1H3MAPTRORC
SCHEMBL1704542 0.80 PKM (0.50) ALDH1A1
SCHEMBL5928658 0.74 CTSD (0.48) CTSDBACE1BACE2
SCHEMBL23059913 0.72 ALDH1A1 (0.48) L3MBTL1TACR1MAPTALDH1A1TSHR
SCHEMBL25643314 0.72 ALDH1A1 (0.48) L3MBTL1TACR1MAPTALDH1A1TSHR
SCHEMBL28296744 0.71 PKM (0.37) L3MBTL1ALDH1A1TSHR
SCHEMBL20679722 0.71 TACR1 (0.34) L3MBTL1TACR1MAPTRORCP2RX1
SCHEMBL12313353 0.71 NR1H3 (0.50) NR1H3MAPTALDH1A1TSHRRORC
SCHEMBL16710463 0.71 ALDH1A1 (0.46) L3MBTL1TACR1MAPTALDH1A1TSHR
SCHEMBL23044998 0.69 ALDH1A1 (0.44) L3MBTL1TACR1MAPTALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0739336-A1 GEM-DISUBSTITUTED AZACYCLIC TACHYKININ ANTAGONISTS MERCK SHARP & DOHME LTD. (GB) 1996-10-30 EP disclosed