SCHEMBL9052744

SCHEMBL9052744

CCCC(=O)c1ccc(N2CCC(O)(c3ccc(C(F)(F)F)cc3)CC2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 10/20 0.59
CYP3A4 P08684 3/20 0.45
CYP2D6 P10635 3/20 0.45
ABCB11 O95342 2/20 0.45
TSHR P16473 2/20 0.45
THPO P40225 2/20 0.45
MTOR P42345 2/20 0.45
EBP Q15125 2/20 0.45
SIGMAR1 Q99720 2/20 0.45
TP53 P04637 1/20 0.45
PKM P14618 1/20 0.45
MAPK1 P28482 1/20 0.45
PMP22 Q01453 2/20 0.45
OPRL1 P41146 1/20 0.45
KDM4E B2RXH2 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HRH3 Q9Y5N1 2/20 0.44
ADRA1A P35348 3/20 0.44
DRD3 P35462 3/20 0.43
DRD4 P21917 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9052324 0.87 DRD2 (0.61) DRD2CYP3A4CYP2D6ABCB11TSHR
SCHEMBL9053341 0.87 ABCB11 (0.62) DRD2CYP3A4CYP2D6ABCB11TSHR
SCHEMBL9050720 0.86 DRD2 (0.57) DRD2CYP3A4CYP2D6ABCB11TSHR
SCHEMBL9053113 0.85 DRD2 (0.56) DRD2CYP3A4CYP2D6KDM4ESMN1; SMN2
SCHEMBL9052696 0.85 DRD2 (0.46) DRD2CYP3A4CYP2D6ABCB11TSHR
SCHEMBL9050732 0.85 DRD2 (0.61) DRD2CYP3A4CYP2D6ABCB11TSHR
SCHEMBL8986025 0.84 DRD2 (0.56) DRD2OPRL1SMN1; SMN2ADRA1AHTR1A
SCHEMBL9052266 0.83 MEN1 (0.58) CYP3A4SIGMAR1SMN1; SMN2HTR1AMEN1
SCHEMBL9052350 0.81 KMT2A (0.53) DRD2SMN1; SMN2ADRA1AHTR1AMEN1
SCHEMBL9052131 0.80 DRD2 (0.42) DRD2CYP3A4CYP2D6ABCB11TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996002250-A1 HALOPERIDOL ANALOGS AND THE USE THEREOF ACEA PHARMACEUTICALS INC. (US) 1996-02-01 WO disclosed