SCHEMBL9052843

SCHEMBL9052843

CN1CCN(c2cccc3ccc(Nc4cccc(C#N)c4)cc23)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.49
HTR1D P28221 4/20 0.49
HTR1B P28222 4/20 0.49
TNIK Q9UKE5 2/20 0.48
KCNH2 Q12809 1/20 0.48
HTR6 P50406 1/20 0.45
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 1/20 0.43
TSHR P16473 1/20 0.43
HRH4 Q9H3N8 1/20 0.42
HRH3 Q9Y5N1 1/20 0.41
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
KMT2A Q03164 1/20 0.40
HIF1A Q16665 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
DRD2 P14416 1/20 0.40
CCNA2 P20248 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6305578 0.82 MAPK14 (0.57) HTR1AHTR1DHTR1BALDH1A1DRD2
SCHEMBL9053159 0.75 WDR5 (0.48) HTR1AHTR1DHTR1BHTR6ALDH1A1
SCHEMBL6305476 0.73 HTR1A (0.54) HTR1AHTR1DHTR1BKCNH2HTR6
SCHEMBL6313054 0.73 MAPT (0.61) HTR1AHTR1DHTR1BKCNH2HTR6
SCHEMBL6308893 0.73 HTR1A (0.50) HTR1AHTR1DHTR1BKCNH2CYP1A2
SCHEMBL6393026 0.72 HTR1A (0.52) HTR1AHTR1DHTR1BCYP1A2ALDH1A1
SCHEMBL6308250 0.72 HTR1A (0.49) HTR1AHTR1DHTR1BCDK2
SCHEMBL8115641 0.72 MAPK14 (0.49) HTR1AHTR1DHTR1BTNIKKCNH2
SCHEMBL6308472 0.71 HTR1A (0.54) HTR1AHTR1DHTR1BHTR6HRH4
SCHEMBL6313298 0.71 HTR1A (0.63) HTR1AHTR1DHTR1BCYP1A2HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0689536-A1 NAPHTHALENE DERIVATIVES PFIZER INC. (US) 1996-01-03 EP disclosed