SCHEMBL9053280

SCHEMBL9053280

CN1CCN(CCc2ccc[c]c2C(N)=O)CC1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
SIGMAR1 Q99720 5/20 0.39
KCNH2 Q12809 2/20 0.38
HRH3 Q9Y5N1 2/20 0.37
ALDH1A1 P00352 1/20 0.35
NAMPT P43490 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
POLB P06746 1/20 0.35
TSHR P16473 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559007 0.89 HRH3 (0.49) HTR2AHTR2CHTR2BSIGMAR1KCNH2
SCHEMBL8554289 0.88 HRH3 (0.48) HTR2AHTR2CHTR2BSIGMAR1HRH3
SCHEMBL9052181 0.85 ALDH1A1 (0.42) SIGMAR1ALDH1A1SMN1; SMN2POLB
SCHEMBL11341667 0.77 SIGMAR1 (0.46) HTR2AHTR2CHTR2BSIGMAR1KCNH2
SCHEMBL8756083 0.73 TAAR1 (0.41) HTR2AHTR2CHTR2BHRH3
SCHEMBL8559413 0.72 HTR2A (0.43) HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL8752394 0.70 HTR1A (0.36) HRH3ALDH1A1TSHRCYP1A2CYP2D6
SCHEMBL28127612 0.69 KDM4E (0.39) HTR2AHTR2CALDH1A1SMN1; SMN2HDAC8
SCHEMBL28626341 0.68 SIGMAR1 (0.53) SIGMAR1HRH3CYP1A2CYP2D6TMEM97
SCHEMBL27907398 0.68 SIGMAR1 (0.67) HTR2AHTR2CHTR2BSIGMAR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996039393-A1 METHOD FOR PREPARING N, N'-DISUBSTITUED CYCLIC UREAS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-12-12 WO claimed
WO-1996000708-A1 METHOD FOR PREPARING ALKYLATING AGENTS AND THEIR USE FOR ALKYLATING CYCLIC UREAS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-01-11 WO claimed
WO-1996039393-A1 METHOD FOR PREPARING N, N'-DISUBSTITUED CYCLIC UREAS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-12-12 WO disclosed
WO-1996000708-A1 METHOD FOR PREPARING ALKYLATING AGENTS AND THEIR USE FOR ALKYLATING CYCLIC UREAS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-01-11 WO disclosed