SCHEMBL9053482

SCHEMBL9053482

O=C1c2ccccc2C(=O)N1CC(F)(F)COC1CCCCO1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
ALDH1A1 P00352 6/20 0.38
KDM4E B2RXH2 1/20 0.38
KDM4C Q9H3R0 1/20 0.37
LMNA P02545 1/20 0.37
KMT2A Q03164 4/20 0.37
TDP1 Q9NUW8 1/20 0.37
HPGD P15428 3/20 0.36
HSD17B10 Q99714 3/20 0.36
MAPT P10636 1/20 0.36
PKM P14618 1/20 0.36
ALOX15 P16050 1/20 0.36
ALOX12 P18054 1/20 0.36
MC4R P32245 1/20 0.36
ACHE P22303 1/20 0.36
MAPK1 P28482 2/20 0.36
MEN1 O00255 2/20 0.36
TSHR P16473 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6473079 0.79 CYP1A2 (0.45) CYP1A2CYP2C9CYP2C19ALDH1A1KDM4E
SCHEMBL6387778 0.77 LMNA (0.43) CYP1A2CYP2C9CYP2C19ALDH1A1KDM4E
SCHEMBL6390234 0.76 HTR1A (0.43) CYP1A2CYP2C9CYP2C19ALDH1A1KDM4E
SCHEMBL28910814 0.76 CYP1A2 (0.47) CYP1A2CYP2C9CYP2C19ALDH1A1KDM4C
SCHEMBL20548002 0.76 CYP1A2 (0.47) CYP1A2CYP2C9CYP2C19ALDH1A1KDM4C
SCHEMBL9053966 0.76 CYP1A2 (0.47) CYP1A2CYP2C9CYP2C19ALDH1A1KDM4E
SCHEMBL29929381 0.76 CYP1A2 (0.47) CYP1A2CYP2C9CYP2C19ALDH1A1KDM4C
SCHEMBL20547967 0.76 CYP1A2 (0.47) CYP1A2CYP2C9CYP2C19ALDH1A1KDM4C
SCHEMBL9053957 0.76 CYP1A2 (0.47) CYP1A2CYP2C9CYP2C19ALDH1A1KDM4E
SCHEMBL22918459 0.75 CYP1A2 (0.49) CYP1A2CYP2C9CYP2C19ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0472181-B1 5-Amine substituted adenosine analogs as immunosuppressants MERRELL PHARMA INC (US) 1996-10-02 EP disclosed
US-5416076-A S-adenosyl methionine decarboxylase inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1995-05-16 US disclosed
US-5308837-A 5'-amine substituted adenosine analogs as immunosuppressants MERRELL DOW PHARMACEUTICALS INC. (US) 1994-05-03 US disclosed
EP-0472181-A2 5-Amine substituted adenosine analogs as immunosuppressants MERRELL PHARMACEUTICALS INC. (US) 1992-02-26 EP disclosed
EP-0358536-A2 Novel S-adenosyl methionine decarboxylase inhibitors MERRELL PHARMACEUTICALS INC. (US) 1990-03-14 EP disclosed
EP-0351475-A1 S-Adenosylmethionine decarboxylase inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1990-01-24 EP disclosed