SCHEMBL9053646

SCHEMBL9053646

Cn1ccc2cc3c(cc21)CCN3C(=O)Nc1cccc(C(F)(F)F)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.67
HTR2A P28223 7/20 0.67
HTR2B P41595 3/20 0.67
CYP1A2 P05177 3/20 0.67
MAPT P10636 2/20 0.67
NPC1 O15118 2/20 0.67
RAB9A P51151 2/20 0.67
PKM P14618 2/20 0.67
KDM4E B2RXH2 1/20 0.67
MEN1 O00255 1/20 0.67
TP53 P04637 1/20 0.67
CYP3A4 P08684 1/20 0.67
CYP2D6 P10635 1/20 0.67
MAPK1 P28482 1/20 0.67
CHRNA7 P36544 1/20 0.67
THPO P40225 1/20 0.67
KMT2A Q03164 1/20 0.67
HIF1A Q16665 1/20 0.67
HDAC6 Q9UBN7 1/20 0.67
SMN1; SMN2 Q16637 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9051246 0.85 HTR2C (0.70) HTR2CHTR2AHTR2BCYP1A2MAPT
SCHEMBL9051316 0.84 RAB9A (0.69) HTR2CHTR2AHTR2BCYP1A2MAPT
SCHEMBL9056673 0.83 HTR2C (0.57) HTR2CHTR2AHTR2BCYP1A2MAPT
SCHEMBL9052878 0.83 NPC1 (0.68) HTR2CHTR2AHTR2BCYP1A2MAPT
SCHEMBL9052562 0.83 NPC1 (0.68) HTR2CHTR2AHTR2BCYP1A2MAPT
SCHEMBL9116372 0.83 HTR2C (0.68) HTR2CHTR2AHTR2BCYP1A2MAPT
SCHEMBL9052182 0.81 MAPT (0.62) HTR2CHTR2AHTR2BCYP1A2MAPT
SCHEMBL29369443 0.80 HTR2C (1.00) HTR2CHTR2AHTR2BCYP1A2MAPT
SCHEMBL1459242 0.80 HTR2C (1.00) HTR2CHTR2AHTR2BCYP1A2MAPT
SCHEMBL29462346 0.80 HTR2C (1.00) HTR2CHTR2AHTR2BCYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0743946-A1 5HT2B RECEPTOR ANTAGONISTS CONDENSED INDOLES SMITHKLINE BEECHAM PLC (GB) 1996-11-27 EP disclosed
WO-1995021844-A1 5HT2B RECEPTOR ANTAGONISTS CONDENSED INDOLES SMITHKLINE BEECHAM PLC (GB) 1995-08-17 WO disclosed