SCHEMBL9054444

SCHEMBL9054444

Cc1cc(CCC(=O)O)ccc1N1CCN(c2nc3c(s2)CCN(C)CC3)C1=O

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.39
S1PR1 P21453 6/20 0.36
DVL1 O14640 1/20 0.36
SLC22A12 Q96S37 2/20 0.34
S1PR5 Q9H228 1/20 0.34
SCD O00767 4/20 0.33
PIM2 Q9P1W9 1/20 0.33
HTR7 P34969 1/20 0.33
FFAR4 Q5NUL3 2/20 0.32
FFAR1 O14842 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
F10 P00742 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9053560 0.90 ALOX15 (0.38) ALOX15S1PR1DVL1SCDPIM2
SCHEMBL7282936 0.69 S1PR1 (0.46) S1PR1SLC22A12FFAR4FFAR1KDM4E
SCHEMBL7274869 0.68 ITGB3 (0.57) S1PR1F10
Hydrochloric Acid SCHEMBL9054174 0.66 DVL1 (0.43) ALOX15DVL1PIM2FFAR4FFAR1
Hydrochloric Acid SCHEMBL7394308 0.65 ITGB3 (0.43) S1PR1
SCHEMBL8559863 0.65 S1PR1 (0.50) S1PR1FFAR1ALDH1A1
SCHEMBL7274574 0.64 ITGB3 (0.57) S1PR1F10
Hydrochloric Acid SCHEMBL8563445 0.64 S1PR1 (0.49) S1PR1FFAR1ALDH1A1
SCHEMBL8559326 0.62 S1PR1 (0.47) S1PR1ALDH1A1F10
SCHEMBL3300620 0.61 F10 (0.40) KDM4EALDH1A1MAPTF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996004271-A1 CONDENSED AZEPINE DERIVATIVES, DRUGS CONTAINING THESE COMPOUNDS AND METHODS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-02-15 WO disclosed