SCHEMBL9054866

SCHEMBL9054866

Cc1ccc(C#N)c2c([N+](=O)[O-])ccc(N(C)Cc3ccncc3)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 7/20 0.47
POLB P06746 2/20 0.40
PIK3CD O00329 1/20 0.39
PIK3R1 P27986 1/20 0.39
PIK3CB P42338 1/20 0.39
TP53 P04637 1/20 0.35
MAPT P10636 3/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
GAA P10253 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
LMNA P02545 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9056780 0.88 TYMS (0.50) TYMSPOLBPIK3CDPIK3R1PIK3CB
SCHEMBL9055262 0.83 TYMS (0.47) TYMSPOLBPIK3CDPIK3R1PIK3CB
SCHEMBL9055802 0.73 TYMS (0.52) TYMSMAPTMEN1CYP2D6CYP2C9
SCHEMBL9056098 0.72 TYMS (0.50) TYMSPOLBPIK3CDPIK3R1PIK3CB
SCHEMBL9054862 0.70 POLB (0.40) POLBTP53MAPTMEN1GAA
SCHEMBL9054766 0.70 VCAM1 (0.42) POLBMAPTMEN1CYP3A4KMT2A
SCHEMBL9055031 0.70 VCAM1 (0.49) POLBMAPTCYP3A4ALDH1A1
SCHEMBL9055527 0.69 TYMS (0.54) TYMSPOLBMAPTMEN1GAA
SCHEMBL9055010 0.65 HTT (0.51) POLBMAPTHTTKMT2ASMN1; SMN2
SCHEMBL9054893 0.64 TYMS (1.00) TYMSMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5545744-A Cyano naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-08-13 US disclosed
US-5498727-A Preparation of benzindole compounds from naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-03-12 US disclosed
WO-1996002502-A1 PREPARATION OF BENZINDOLE COMPOUNDS FROM NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1996-02-01 WO disclosed