SCHEMBL9056780

SCHEMBL9056780

Cc1cc(CN(C)c2ccc([N+](=O)[O-])c3c(C#N)ccc(C)c23)ccn1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TYMS P04818 6/20 0.50
MAPT P10636 2/20 0.35
CTSB P07858 1/20 0.35
POLB P06746 2/20 0.33
ALDH1A1 P00352 1/20 0.33
GRM5 P41594 1/20 0.32
PIK3CD O00329 1/20 0.32
PIK3R1 P27986 1/20 0.32
PIK3CB P42338 1/20 0.32
VCAM1 P19320 1/20 0.32
CDK4 P11802 1/20 0.32
CDK2 P24941 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9054866 0.88 TYMS (0.47) TYMSMAPTPOLBALDH1A1PIK3CD
SCHEMBL9055802 0.85 TYMS (0.52) TYMSMAPTCTSBALDH1A1
SCHEMBL9055527 0.74 TYMS (0.54) TYMSMAPTCTSBPOLBALDH1A1
SCHEMBL9055262 0.71 TYMS (0.47) TYMSMAPTCTSBPOLBALDH1A1
SCHEMBL9056098 0.69 TYMS (0.50) TYMSMAPTCTSBPOLBALDH1A1
SCHEMBL9055272 0.69 CTSB (0.40) MAPTCTSBALDH1A1LMNA
SCHEMBL9055031 0.67 VCAM1 (0.49) MAPTPOLBALDH1A1VCAM1
SCHEMBL9054766 0.67 VCAM1 (0.42) MAPTPOLBALDH1A1VCAM1LMNA
SCHEMBL9055086 0.67 TYMS (1.00) TYMS
SCHEMBL8103078 0.62 MEN1 (0.40) MAPTCTSBPOLBALDH1A1VCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5545744-A Cyano naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-08-13 US disclosed
US-5498727-A Preparation of benzindole compounds from naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-03-12 US disclosed
WO-1996002502-A1 PREPARATION OF BENZINDOLE COMPOUNDS FROM NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1996-02-01 WO disclosed