SCHEMBL9055262

SCHEMBL9055262

CN(Cc1ccncc1)c1ccc([N+](=O)[O-])c2c(C#N)cccc12

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TYMS P04818 9/20 0.47
POLB P06746 1/20 0.42
CTSB P07858 2/20 0.39
PIK3CD O00329 1/20 0.39
PIK3R1 P27986 1/20 0.39
PIK3CB P42338 1/20 0.39
MAPT P10636 3/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPK1 P28482 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
LRRK2 Q5S007 1/20 0.38
TP53 P04637 1/20 0.36
LMNA P02545 1/20 0.35
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9056098 0.89 TYMS (0.50) TYMSPOLBCTSBPIK3CDPIK3R1
SCHEMBL9055802 0.87 TYMS (0.52) TYMSCTSBMAPTALDH1A1MAPK1
SCHEMBL9055527 0.85 TYMS (0.54) TYMSPOLBCTSBMAPTALDH1A1
SCHEMBL9054866 0.83 TYMS (0.47) TYMSPOLBPIK3CDPIK3R1PIK3CB
SCHEMBL9054758 0.72 HTR6 (0.48) ALDH1A1MAPK1LMNA
SCHEMBL9056780 0.71 TYMS (0.50) TYMSPOLBCTSBPIK3CDPIK3R1
SCHEMBL9508662 0.71 TYMS (0.59) TYMSPOLBMAPTALDH1A1MAPK1
SCHEMBL9055252 0.70 POLB (0.42) POLBCTSBMAPTALDH1A1MAPK1
SCHEMBL11811062 0.69 TDP1 (0.55) POLBCTSBMAPTALDH1A1GAA
SCHEMBL9055020 0.69 TDP1 (0.42) POLBCTSBMAPTALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5545744-A Cyano naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-08-13 US disclosed
US-5498727-A Preparation of benzindole compounds from naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-03-12 US disclosed
WO-1996002502-A1 PREPARATION OF BENZINDOLE COMPOUNDS FROM NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1996-02-01 WO disclosed