SCHEMBL9054968

SCHEMBL9054968

FC(F)(F)c1cccc(Cn2cc(CCNc3ccncc3)c3ccccc32)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.50
YES1 P07947 1/20 0.47
KDR P35968 1/20 0.47
JAK3 P52333 1/20 0.47
HTR2C P28335 1/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
GAA P10253 1/20 0.45
CYP2D6 P10635 1/20 0.45
MAPT P10636 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
PARP1 P09874 1/20 0.44
ICMT O60725 7/20 0.43
CYP19A1 P11511 4/20 0.43
CHEK1 O14757 1/20 0.43
DAPK3 O43293 1/20 0.43
ROCK2 O75116 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8416389 0.86 HTR2C (0.59) HTR6YES1KDRJAK3HTR2C
SCHEMBL8806145 0.82 YES1 (0.55) YES1KDRJAK3ALDH1A1GAA
SCHEMBL8418190 0.81 CYP19A1 (0.58) HTR6YES1KDRJAK3HTR2C
SCHEMBL9055307 0.81 YES1 (0.69) HTR6YES1KDRJAK3HTR2C
SCHEMBL16026993 0.80 HTR6 (0.55) HTR6KDRALDH1A1CYP1A2CYP3A4
SCHEMBL4354844 0.79 ICMT (0.54) HTR6ALDH1A1CYP1A2CYP3A4GAA
SCHEMBL9056608 0.77 CYP19A1 (0.55) YES1KDRJAK3HTR2CALDH1A1
SCHEMBL24144381 0.75 ICMT (0.50) HTR6KDRICMTROCK2ROCK1
SCHEMBL8418107 0.74 CYP19A1 (0.56) HTR6YES1KDRJAK3HTR2C
SCHEMBL24143255 0.74 NR1D1 (0.47) HTR6ICMTROCK2ROCK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996004266-A2 INDOL, INDAZOL, PYRIDOPYRROL AND PYRIDOPYRAZOL DERIVATIVES WITH ANTI-ASTHMATIC, ANTI-ALLERGIC, ANTI-INFLAMMATORY AND IMMUNOMODULATING EFFECTS ASTA MEDICA AKTIENGESELLSCHAFT (DE) 1996-02-15 WO disclosed