SCHEMBL9055189

SCHEMBL9055189

CN(Cc1cccc2c1ccn2S(=O)(=O)c1ccccc1)c1ccc2c3c(cccc13)C(N)=N2

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TYMS P04818 9/20 0.61
HTR6 P50406 11/20 0.53
HTR1A P08908 2/20 0.53
HTR1D P28221 2/20 0.53
HTR1B P28222 2/20 0.53
HTR1F P30939 2/20 0.53
HTR7 P34969 2/20 0.53
DRD3 P35462 2/20 0.53
DRD2 P14416 2/20 0.53
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
HTR2A P28223 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3622409 0.76 HTR6 (0.77) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL9054758 0.73 HTR6 (0.48) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL4029770 0.71 HTR6 (0.72) HTR6HTR1AHTR1DHTR1BHTR1F
Metesind SCHEMBL6703943 0.70 TYMS (1.00) TYMS
SCHEMBL7449413 0.70 HTR6 (0.71) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL3611374 0.70 HTR6 (0.80) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL7245193 0.70 HTR6 (1.00) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL13378917 0.69 HTR6 (0.66) HTR6HTR1AHTR1DHTR1BHTR1F
Hydrochloric Acid SCHEMBL3624923 0.69 HTR6 (0.78) HTR6HTR1AHTR1DHTR1BHTR1F
Trifluoroacetic Acid SCHEMBL3621161 0.69 HTR6 (0.65) HTR6HTR1AHTR1DHTR1BHTR1F

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5545744-A Cyano naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-08-13 US disclosed
US-5498727-A Preparation of benzindole compounds from naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-03-12 US disclosed
WO-1996002502-A1 PREPARATION OF BENZINDOLE COMPOUNDS FROM NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1996-02-01 WO disclosed