SCHEMBL9054758

SCHEMBL9054758

CN(Cc1cccc2c1ccn2S(=O)(=O)c1ccccc1)c1ccc([N+](=O)[O-])c2c(C#N)cccc12

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 19/20 0.48
HTR1A P08908 3/20 0.48
HTR1D P28221 3/20 0.48
HTR1B P28222 3/20 0.48
HTR1F P30939 3/20 0.48
HTR7 P34969 3/20 0.48
DRD3 P35462 3/20 0.48
DRD2 P14416 2/20 0.48
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
HTR2A P28223 1/20 0.40
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3622409 0.73 HTR6 (0.77) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL9055189 0.73 TYMS (0.61) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL9055262 0.72 TYMS (0.47) ALDH1A1LMNAMAPK1
SCHEMBL4785680 0.71 HTR6 (0.62) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL29687030 0.70 HTR6 (0.61) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL3241536 0.70 HTR6 (0.61) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL9056098 0.70 TYMS (0.50) ALDH1A1LMNAMAPK1
SCHEMBL9055802 0.69 TYMS (0.52) CYP2D6ALDH1A1MAPK1SMN1; SMN2
SCHEMBL4029770 0.68 HTR6 (0.72) HTR6HTR1AHTR1DHTR1BHTR1F
SCHEMBL9508662 0.68 TYMS (0.59) ALDH1A1LMNAMAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5545744-A Cyano naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-08-13 US disclosed
US-5498727-A Preparation of benzindole compounds from naphthalene compounds AGOURON PHARMACEUTICALS, INC. (US) 1996-03-12 US disclosed
WO-1996002502-A1 PREPARATION OF BENZINDOLE COMPOUNDS FROM NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1996-02-01 WO disclosed