SCHEMBL9055658

SCHEMBL9055658

COC(=O)C1CC(C#N)(c2ccccc2F)CCC1=O.COC(=O)CCC(C#N)(CCC(=O)OC)c1ccccc1F

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.37
PSEN2 P49810 1/20 0.37
APH1B Q8WW43 1/20 0.37
NCSTN Q92542 1/20 0.37
APH1A Q96BI3 1/20 0.37
PSENEN Q9NZ42 1/20 0.37
RORC P51449 1/20 0.35
ADRA1D P25100 2/20 0.33
ADRA1A P35348 2/20 0.33
ADRA1B P35368 2/20 0.33
BDKRB1 P46663 1/20 0.32
PKM P14618 1/20 0.31
ALDH1A1 P00352 1/20 0.31
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8356325 0.85 PSEN1 (0.46) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL11920949 0.78 ALDH1A1 (0.39) PKMALDH1A1
SCHEMBL8022068 0.75 ADRA1A (0.39) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL11088958 0.75 PSEN1 (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL11826260 0.75 PSEN1 (0.37) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL735539 0.74 MEN1 (0.42) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4430870 0.73 PSEN1 (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL11822928 0.73 MAPT (0.38) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1558214 0.72 RORC (0.45) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL17542850 0.72 PSEN1 (0.52) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996011934-A1 TRICYCLIC SPIRO COMPOUNDS PROCESS FOR THEIR PREPARATION AND THEIR USE AS 5HT1D RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-04-25 WO disclosed