SCHEMBL9056097

SCHEMBL9056097

COc1ccc2c(C(=O)c3ccccc3O)c(-c3ccccc3OC)oc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.50
ALOX15 P16050 3/20 0.50
HPGD P15428 3/20 0.50
AR P10275 2/20 0.50
CYP1A2 P05177 2/20 0.50
CYP2C19 P33261 2/20 0.50
LMNA P02545 1/20 0.50
PGR P06401 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
CHRM1 P11229 1/20 0.50
TBXA2R P21731 1/20 0.50
SLC6A2 P23975 1/20 0.50
ADRA1A P35348 1/20 0.50
HIF1A Q16665 1/20 0.50
ALOX5 P09917 2/20 0.47
KDM4E B2RXH2 4/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
TSHR P16473 2/20 0.47
HTT P42858 1/20 0.47
MEN1 O00255 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8745272 0.86 SLC22A12 (0.60) CYP3A4ALOX15HPGDARCYP2C19
SCHEMBL15864338 0.79 ALOX5 (0.70) HPGDALOX5KDM4ETSHRMEN1
SCHEMBL5138931 0.78 KDM4E (0.74) CYP3A4ALOX15HPGDCYP1A2CYP2C19
SCHEMBL15865400 0.72 AR (0.47) CYP3A4ALOX15HPGDARCYP1A2
SCHEMBL7332022 0.71 CYP3A4 (0.62) CYP3A4ALOX15HPGDARCYP1A2
SCHEMBL5433434 0.71 KDM4E (0.74) CYP3A4ALOX15HPGDARCYP2C19
SCHEMBL1874869 0.70 HPGD (0.79) CYP3A4ALOX15HPGDARCYP1A2
SCHEMBL15864329 0.70 KDM4E (0.64) CYP3A4ALOX15HPGDCYP2C19LMNA
SCHEMBL17270585 0.70 KDM4E (0.57) HPGDLMNAADORA3ALOX5KDM4E
SCHEMBL6426148 0.69 TUBB4A (0.63) CYP3A4ALOX15ADORA3SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996012489-A1 BICYCLIC NEUROPEPTIDE Y RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1996-05-02 WO disclosed