SCHEMBL9056243

SCHEMBL9056243

O=C(O)Oc1cn(-c2ccc(CN3CCOCC3)cc2)c2c(Cl)c(F)c(F)cc2c1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 1/20 0.40
MAPK9 P45984 1/20 0.40
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
TP53 P04637 2/20 0.40
KCNH2 Q12809 4/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
HSP90AA1 P07900 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
POLA1 P09884 2/20 0.38
PIK3CD O00329 1/20 0.38
PIK3R2 O00459 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
PIK3CG P48736 1/20 0.38
PIK3R5 Q8WYR1 1/20 0.38
PIK3R3 Q92569 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9056238 0.89 ALDH1A1 (0.50) NPC1RAB9ASMN1; SMN2TP53KCNH2
SCHEMBL8801306 0.82 PIM1 (0.37) MAPK8SMN1; SMN2ALDH1A1KDM4EPOLB
SCHEMBL9048087 0.82 KDM4E (0.41) MAPK8SMN1; SMN2KCNH2ALDH1A1KDM4E
SCHEMBL9055113 0.81 MAPK8 (0.51) MAPK8MAPK9NPC1RAB9ASMN1; SMN2
SCHEMBL9056323 0.81 PIM1 (0.37) MAPK8SMN1; SMN2KCNH2ALDH1A1KDM4E
SCHEMBL8801570 0.79 PIM1 (0.37) MAPK8ALDH1A1KDM4EPOLBHSP90AA1
SCHEMBL8803705 0.79 HDAC1 (0.38) ALDH1A1KDM4EPOLBHSP90AA1RXFP1
SCHEMBL9043747 0.77 TOP1 (0.51) ALDH1A1KDM4EPOLBHSP90AA1RXFP1
SCHEMBL8801060 0.76 TOP1 (0.39) SMN1; SMN2TP53ALDH1A1KDM4EPOLB
SCHEMBL9055563 0.76 MAPK8 (0.37) MAPK8SMN1; SMN2ALDH1A1KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996002510-A1 NOVEL 1-[4(AMINO METHYL)PHENYL] SUBSTITUTED QUINOLONE CARBOXYLIC ACIDS BAYER AKTIENGESELLSCHAFT (DE) 1996-02-01 WO disclosed