SCHEMBL9056601

SCHEMBL9056601

CCOC(=O)CN(C(=O)[C@H](CCC(N)c1ncc[nH]1)NS(=O)(=O)c1cccc2cc(C)cnc12)C1CC1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC16A3 O15427 1/20 0.34
SLC40A1 Q9NP59 6/20 0.33
HTR6 P50406 1/20 0.33
ALDH1A1 P00352 2/20 0.33
PDE2A O00408 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
P2RY12 Q9H244 1/20 0.32
F2 P00734 1/20 0.31
PKLR P30613 1/20 0.31
PARP1 P09874 1/20 0.31
ALOX15 P16050 1/20 0.31
MAPK1 P28482 1/20 0.31
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9056228 0.84 ITGB3 (0.41) ALDH1A1PDE2APDE3BPDE3AP2RY12
SCHEMBL9055326 0.84 ITGB3 (0.40) ALDH1A1PDE2APDE3BPDE3AP2RY12
SCHEMBL9056960 0.83 ITGB3 (0.40) PDE2APDE3BPDE3AP2RY12F2
SCHEMBL8716492 0.83 SLC16A3 (0.37) SLC16A3SLC40A1HTR6ALDH1A1F2
SCHEMBL7324729 0.81 HTR6 (0.36) SLC16A3SLC40A1HTR6ALDH1A1F2
SCHEMBL9054354 0.80 CCR10 (0.40)
SCHEMBL9055303 0.78 ITGB3 (0.44) SLC16A3
SCHEMBL9056174 0.77 F2 (0.41) F2
SCHEMBL9054627 0.77 CCR10 (0.39) PDE2APDE3BPDE3AP2RY12
SCHEMBL9056911 0.75 ITGB3 (0.41) SLC16A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996002517-A1 SUBSTITUTED ARYLSULFONAMIDES, THEIR PREPARATION AND USE AS THROMBIN-INHIBITING MEDICAMENTS DR. KARL THOMAE GMBH (DE) 1996-02-01 WO disclosed