SCHEMBL9057638

SCHEMBL9057638

Cc1cc(C)c(NC(=O)N(Cc2ccc(-c3c[nH]nc3C)cc2)C2CCCCCC2)c(C)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ALDH1A1 P00352 6/20 0.39
KDM4E B2RXH2 5/20 0.39
NPC1 O15118 1/20 0.39
ROCK2 O75116 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
LTB4R2 Q9NPC1 1/20 0.38
TP53 P04637 3/20 0.37
MAPT P10636 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
POLB P06746 1/20 0.36
HSD17B10 Q99714 3/20 0.36
UBE2M P61081 1/20 0.36
DCUN1D1 Q96GG9 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8810366 0.84 ROCK2 (0.55) GAANPSR1ROCK2
SCHEMBL8814244 0.84 GAA (0.44) GAANPSR1ALDH1A1KDM4ENPC1
SCHEMBL8809779 0.84 GAA (0.52) GAANPSR1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL9056512 0.84 KDM4E (0.36) GAANPSR1ALDH1A1KDM4ENPC1
SCHEMBL9056936 0.82 GAA (0.50) GAANPSR1ALDH1A1SMN1; SMN2LTB4R2
SCHEMBL8817897 0.82 GAA (0.47) GAANPSR1ALDH1A1KDM4EROCK2
SCHEMBL8817749 0.81 NPSR1 (0.49) GAANPSR1ALDH1A1SMN1; SMN2TP53
SCHEMBL8807180 0.81 GAA (0.49) GAANPSR1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL8808422 0.81 TP53 (0.52) GAANPSR1ALDH1A1TP53POLB
SCHEMBL8817744 0.81 NPSR1 (0.45) GAANPSR1ALDH1A1SMN1; SMN2LTB4R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996010559-A1 UREA DERIVATIVES AND THEIR USE AS ACAT-INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-04-11 WO disclosed