SCHEMBL9056512

SCHEMBL9056512

CSc1cc(C)nc(SC)c1NC(=O)N(Cc1ccc(-c2c[nH]nc2C)cc1)C1CCCCCC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.36
ALDH1A1 P00352 5/20 0.36
NPC1 O15118 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
USP2 O75604 3/20 0.34
HPGD P15428 2/20 0.34
HSD17B10 Q99714 2/20 0.34
ROCK2 O75116 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
SOAT1 P35610 5/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
LTB4R2 Q9NPC1 1/20 0.34
NPSR1 Q6W5P4 2/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8817633 0.92 ROCK2 (0.38) KDM4EALDH1A1NPC1CYP1A2CYP3A4
SCHEMBL8344843 0.86 KDM4E (0.42) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL9057638 0.84 GAA (0.43) KDM4EALDH1A1NPC1CYP1A2CYP3A4
SCHEMBL8808860 0.83 USP2 (0.43) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL8856425 0.82 GCGR (0.37) KDM4EALDH1A1NPC1CYP1A2CYP3A4
SCHEMBL8809049 0.82 TP53 (0.42) ALDH1A1CYP1A2CYP2C19USP2NPSR1
SCHEMBL8807728 0.82 TP53 (0.42) ALDH1A1CYP1A2CYP2C19USP2NPSR1
SCHEMBL29972806 0.82 TP53 (0.42) ALDH1A1CYP1A2CYP2C19USP2NPSR1
SCHEMBL9058046 0.82 UBE2M (0.41) KDM4EALDH1A1NPC1CYP1A2CYP3A4
SCHEMBL9056629 0.82 KMT2A (0.38) KDM4EALDH1A1NPC1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996010559-A1 UREA DERIVATIVES AND THEIR USE AS ACAT-INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-04-11 WO disclosed