SCHEMBL9057670

SCHEMBL9057670

CC(C)OC(=O)CCc1ccc(-c2nc(-c3ccc4c(c3)CCN(C(=O)C(F)(F)F)CC4)cs2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DVL1 O14640 1/20 0.41
CDC25A P30304 4/20 0.40
CDC25B P30305 4/20 0.40
CDC25C P30307 4/20 0.40
DUSP3 P51452 4/20 0.40
MAPT P10636 5/20 0.37
SMN1; SMN2 Q16637 5/20 0.37
NPC1 O15118 4/20 0.37
RAB9A P51151 4/20 0.37
ALDH1A1 P00352 4/20 0.37
HPGD P15428 2/20 0.37
ALOX15 P16050 2/20 0.37
HSD17B10 Q99714 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
USP2 O75604 1/20 0.37
TP53 P04637 3/20 0.37
GFER P55789 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9057948 0.75 DVL1 (0.56) DVL1CDC25ACDC25BCDC25CDUSP3
SCHEMBL9063378 0.75 ESR1 (0.41) DVL1NPC1RAB9AHPGDHSD17B10
SCHEMBL9056388 0.69 NPC1 (0.38) MAPTSMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL1364723 0.66 ESR1 (0.52) NPC1RAB9AESR1ESR2MEN1
SCHEMBL16092839 0.66 POLB (0.46) CDC25ACDC25BCDC25CDUSP3MAPT
SCHEMBL31173327 0.65 ESR2 (0.57) ESR1ESR2
SCHEMBL9055466 0.65 ALDH1A1 (0.46) DVL1CDC25ACDC25BCDC25CDUSP3
SCHEMBL4768506 0.64 DRD3 (0.50) ESR1ESR2
SCHEMBL1367276 0.64 ESR1 (0.52) NPC1HPGDCYP3A4CYP2C19ESR1
SCHEMBL8565812 0.64 NOTUM (0.39) MAPTSMN1; SMN2ALDH1A1ALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996004271-A1 CONDENSED AZEPINE DERIVATIVES, DRUGS CONTAINING THESE COMPOUNDS AND METHODS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-02-15 WO disclosed