SCHEMBL9058240

SCHEMBL9058240

CC(C)(C)C(=O)Nc1ccc(C(F)(F)F)cc1C(O)c1cccc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
RXFP1 Q9HBX9 1/20 0.41
ADRA2C P18825 2/20 0.40
SLC6A2 P23975 2/20 0.40
HTR2C P28335 2/20 0.40
SLC6A4 P31645 2/20 0.40
OPRM1 P35372 2/20 0.40
DRD3 P35462 2/20 0.40
CASR P41180 2/20 0.40
MLNR O43193 1/20 0.40
ABCB11 O95342 1/20 0.40
ADRB1 P08588 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
CYP2D6 P10635 1/20 0.40
CHRM1 P11229 1/20 0.40
DRD2 P14416 1/20 0.40
CHRM3 P20309 1/20 0.40
GLRA1 P23415 1/20 0.40
AVPR2 P30518 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4112920 0.80 ALDH1A1 (0.45) ALDH1A1L3MBTL1RXFP1CYP2D6HTT
SCHEMBL8946084 0.71 GAA (0.48) ALDH1A1L3MBTL1HTTTACR1KCNJ11
SCHEMBL12862996 0.70 KDM4E (0.62) ALDH1A1CYP2D6MAPK14HDAC1HDAC7
SCHEMBL13776424 0.70 HSP90AA1 (0.43) ALDH1A1RXFP1MEN1KMT2A
SCHEMBL13015660 0.70 KIF11 (0.52) ALDH1A1L3MBTL1TACR1KCNJ11KDM4E
SCHEMBL4121438 0.69 MEN1 (0.46) ALDH1A1RXFP1TRPV1KDM4EMEN1
SCHEMBL8687043 0.69 HTT (0.52) L3MBTL1CYP2D6HTTTRPV1KCNJ11
SCHEMBL14146416 0.69 RXFP1 (0.47) ALDH1A1L3MBTL1RXFP1ADRA2CADRB1
SCHEMBL14568587 0.69 CFTR (0.51) ALDH1A1L3MBTL1TACR1HDAC1KDM4E
SCHEMBL14146163 0.68 RXFP1 (0.46) ALDH1A1L3MBTL1RXFP1CYP2D6HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996020184-A1 NAPHTHYL-BENZOXAZEPINES OR -BENZOTHIAZEPINES AS SQUALENE SYNTHETASE INHIBITORS PFIZER INC. (US) 1996-07-04 WO disclosed