SCHEMBL9058568

SCHEMBL9058568

O=C(NCCSc1ccc2ncc([N+](=O)[O-])n2n1)C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
HPGD P15428 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
GLA P06280 1/20 0.39
ALOX12 P18054 1/20 0.39
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
GSTO1 P78417 1/20 0.34
IDO1 P14902 1/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C9 P11712 2/20 0.33
KDM4E B2RXH2 2/20 0.32
CYP2C19 P33261 1/20 0.32
HSD17B10 Q99714 1/20 0.32
DYRK3 O43781 1/20 0.31
CCNT1 O60563 1/20 0.31
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
CDK9 P50750 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9058728 0.86 GSTP1 (0.42) ALDH1A1SMN1; SMN2GLARAB9ACYP1A2
SCHEMBL9058779 0.82 CYP1A2 (0.33) ALDH1A1HPGDSMN1; SMN2GLAALOX12
SCHEMBL9058562 0.81 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2MAPTRAB9ACYP1A2
SCHEMBL9058877 0.81 CYP1A2 (0.33) ALDH1A1HPGDCYP1A2CYP2C9KDM4E
SCHEMBL9058881 0.77 KDM4E (0.46) ALDH1A1HPGDSMN1; SMN2RAB9ACYP1A2
SCHEMBL9059134 0.76 GLA (0.37) ALDH1A1HPGDGLAMAPTCYP1A2
SCHEMBL9058693 0.73 MAPK1 (0.43) ALDH1A1GLACYP1A2CYP2C9KDM4E
SCHEMBL9058715 0.72 MKNK1 (0.39) CYP1A2CYP2C9DYRK3CCNT1CCNA2
SCHEMBL9058809 0.72 MKNK1 (0.39) CYP1A2CYP2C9DYRK3CCNT1CCNA2
SCHEMBL9058875 0.72 KDM4E (0.54) ALDH1A1HPGDSMN1; SMN2MAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996016656-A1 CONDENSED IMIDAZOLE DERIVATIVES, THEIR PREPARATION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-06-06 WO disclosed