SCHEMBL9058575

SCHEMBL9058575

O=[C]C(=CNc1ccc(Cn2ccnn2)cc1)C(=O)c1cc(F)c(F)c(F)c1F

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.39
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
F2 P00734 1/20 0.32
F10 P00742 1/20 0.32
KLKB1 P03952 2/20 0.31
ALDH1A1 P00352 1/20 0.31
HSD17B1 P14061 1/20 0.31
HSD17B2 P37059 1/20 0.31
IDO1 P14902 1/20 0.30
TDO2 P48775 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9058577 0.86 CYP19A1 (0.37) CYP19A1F2F10KLKB1ALDH1A1
SCHEMBL8801294 0.82 DHODH (0.43) CYP19A1ALDH1A1
SCHEMBL8802032 0.75 NPSR1 (0.42) ALDH1A1
SCHEMBL9415867 0.72 DHODH (0.44) CYP19A1ALDH1A1
SCHEMBL9415889 0.66 DHODH (0.43) ALDH1A1
SCHEMBL29820189 0.62 CYP19A1 (0.67) CYP19A1ALDH1A1IDO1TDO2
SCHEMBL8801565 0.60 PIM1 (0.47) CYP19A1ALDH1A1
SCHEMBL27927514 0.60 CYP19A1 (0.64) CYP19A1KLKB1ALDH1A1
SCHEMBL10372641 0.60 DHODH (0.54) ALDH1A1
SCHEMBL10372640 0.60 DHODH (0.54) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996002533-A1 NOVEL 6- AND 6,8-SUBSTITUTED 1-[4-(1H-1,2,4-TRIAZOL-1-YL METHYL) PHENYL] QUINOLONE CARBOXYLIC ACIDS BAYER AKTIENGESELLSCHAFT (DE) 1996-02-01 WO disclosed