SCHEMBL9060183

SCHEMBL9060183

CCc1cnc(-c2ccc(-c3ccc(OC(F)F)cc3)cc2)nc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 3/20 0.48
GRIN2B Q13224 3/20 0.48
RXRA P19793 2/20 0.48
DRD1 P21728 1/20 0.42
RAB9A P51151 4/20 0.42
NPC1 O15118 3/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPT P10636 2/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
PTGER4 P35408 1/20 0.40
HDAC4 P56524 2/20 0.38
ALKBH1 Q13686 1/20 0.38
SCN5A Q14524 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.36
TP53 P04637 1/20 0.36
HTT P42858 2/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9061744 0.98 RXRA (0.49) GRIN1GRIN2BRXRADRD1RAB9A
SCHEMBL9060293 0.93 RXRA (0.46) GRIN1GRIN2BRXRADRD1RAB9A
SCHEMBL9060670 0.90 DRD1 (0.44) GRIN1GRIN2BRXRADRD1RAB9A
SCHEMBL9062438 0.88 RAB9A (0.43) GRIN1GRIN2BRXRADRD1RAB9A
SCHEMBL9513537 0.86 RAB9A (0.41) GRIN1GRIN2BRXRARAB9ANPC1
SCHEMBL9062036 0.86 RAB9A (0.44) GRIN1GRIN2BRXRADRD1RAB9A
SCHEMBL9062296 0.85 RARB (0.49) GRIN1GRIN2BRXRADRD1RAB9A
SCHEMBL9062271 0.84 RARB (0.54) DRD1RAB9ANPC1SMN1; SMN2HSD17B10
SCHEMBL9062353 0.84 RARB (0.50) GRIN1GRIN2BRXRADRD1RAB9A
SCHEMBL9061164 0.83 RARB (0.56) RAB9ANPC1SMN1; SMN2HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5536442-A ELECTROOPTICS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-07-16 US disclosed
US-5389292-A Liquid crystalline media having positive dielctric anisotropy, chemical, heat and radiation resistance, used as electro-optical displaying MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-14 US disclosed
EP-0381728-B1 DIFLUOROMETHYL COMPOUNDS MERCK PATENT GMBH (DE) 1993-12-08 EP disclosed