SCHEMBL9060747

SCHEMBL9060747

CCCCc1ccc(CCc2ccc(OC(F)(F)F)cc2)c(F)c1F

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.41
DAO P14920 1/20 0.41
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
SLC6A4 P31645 5/20 0.40
SLC6A3 Q01959 4/20 0.40
GPR84 Q9NQS5 1/20 0.39
ALDH1A1 P00352 1/20 0.38
ALOX5 P09917 1/20 0.38
PPARG P37231 1/20 0.38
FAAH O00519 1/20 0.36
ESR1 P03372 1/20 0.35
CYP19A1 P11511 1/20 0.35
ESR2 Q92731 1/20 0.35
SCN8A Q9UQD0 1/20 0.35
CASR P41180 1/20 0.35
PLA2G4A P47712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9061607 0.96 FAAH (0.41) TSHRDAOHDAC3HDAC1HDAC2
SCHEMBL9061734 0.91 TSHR (0.43) TSHRDAOHDAC3HDAC1HDAC2
SCHEMBL9061433 0.88 DAO (0.46) TSHRDAOSLC6A4SLC6A3GPR84
SCHEMBL9060258 0.88 ALOX5 (0.39) TSHRDAOHDAC3HDAC1HDAC2
SCHEMBL9062396 0.86 TSHR (0.49) TSHRDAOHDAC3HDAC1HDAC2
SCHEMBL9061450 0.86 ALOX5 (0.38) TSHRDAOHDAC3HDAC1HDAC2
SCHEMBL2056243 0.84 TSHR (0.50) TSHRDAOHDAC3HDAC1HDAC2
SCHEMBL9062034 0.83 HDAC3 (0.39) TSHRHDAC3HDAC1HDAC2
SCHEMBL9060352 0.83 HCRTR1 (0.44) TSHRDAO
SCHEMBL10532774 0.83 PPARG (0.39) DAOHDAC3HDAC1HDAC2GPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5536442-A ELECTROOPTICS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1996-07-16 US disclosed
US-5324449-A Substituted phenyl trifluoromethyl ethers MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1994-06-28 US disclosed
EP-0334911-B1 SUBSTITUTED PHENYLTRIFLUORMETHYLETHERS MERCK PATENT GmbH (DE) 1993-02-10 EP disclosed
EP-0334911-A1 SUBSTITUTED PHENYLTRIFLUORMETHYLETHERS MERCK PATENT GmbH (DE) 1989-10-04 EP disclosed
WO-1989002884-A1 SUBSTITUTED PHENYLTRIFLUORMETHYLETHERS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1989-04-06 WO disclosed