SCHEMBL9062121

SCHEMBL9062121

O=C(O)/C=C/c1ccoc1.O=C(O)C=Cc1cccs1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 3/20 0.69
ALDH1A1 P00352 3/20 0.46
MAPT P10636 3/20 0.46
ABCG2 Q9UNQ0 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
LMNA P02545 2/20 0.43
HDAC3 O15379 1/20 0.42
TNKS O95271 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9062123 1.00 HCAR2 (0.69) HCAR2ALDH1A1MAPTABCG2SMN1; SMN2
SCHEMBL660178 0.83 HCAR2 (1.00) HCAR2ALDH1A1MAPTSMN1; SMN2LMNA
SCHEMBL564789 0.83 HCAR2 (1.00) HCAR2ALDH1A1MAPTSMN1; SMN2LMNA
SCHEMBL7893859 0.83 HCAR2 (1.00) HCAR2ALDH1A1MAPTSMN1; SMN2LMNA
SCHEMBL600082 0.83 HCAR2 (1.00) HCAR2ALDH1A1MAPTABCG2SMN1; SMN2
SCHEMBL143282 0.83 HCAR2 (1.00) HCAR2ALDH1A1MAPTABCG2SMN1; SMN2
Hydrochloric Acid SCHEMBL9874572 0.81 HCAR2 (0.96) HCAR2ALDH1A1MAPTABCG2SMN1; SMN2
SCHEMBL4212112 0.81 HCAR2 (0.96) HCAR2ALDH1A1MAPTABCG2SMN1; SMN2
Hydrochloric Acid SCHEMBL9261463 0.81 HCAR2 (0.96) HCAR2ALDH1A1MAPTSMN1; SMN2LMNA
Hydrochloric Acid SCHEMBL27913308 0.81 HCAR2 (0.96) HCAR2ALDH1A1MAPTABCG2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996040732-A1 COMBINATORIAL NON-PEPTIDE LIBRARIES ZYMOGENETICS, INC. (US) 1996-12-19 WO disclosed