SCHEMBL906519

SCHEMBL906519

CC(C)(C)OC(=O)NCCc1cc(Br)cc2[nH]c(=O)c(C(F)(F)F)nc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 1/20 0.43
CACNA1B Q00975 1/20 0.43
CACNA1C Q13936 1/20 0.43
NQO2 P16083 1/20 0.39
BCHE P06276 1/20 0.37
IDO1 P14902 3/20 0.36
KDM4E B2RXH2 6/20 0.36
HSD17B10 Q99714 6/20 0.36
ALDH1A1 P00352 4/20 0.36
TSHR P16473 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
GFER P55789 1/20 0.35
HPGD P15428 2/20 0.34
CYP1A2 P05177 1/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HIF1A Q16665 1/20 0.34
PDE3B Q13370 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL906377 0.87 NQO2 (0.41) CACNA1HCACNA1BCACNA1CNQO2BCHE
SCHEMBL3844306 0.72 IDO1 (0.48) NQO2IDO1KDM4EHSD17B10ALDH1A1
SCHEMBL28801452 0.69 NQO2 (0.47) CACNA1HCACNA1BCACNA1CNQO2IDO1
SCHEMBL7841704 0.67 MTNR1A (0.51) NQO2BCHEKDM4EHSD17B10ALDH1A1
SCHEMBL13400107 0.67 CA1 (0.46) NQO2IDO1KDM4EALDH1A1NPSR1
SCHEMBL30981863 0.67 NQO2 (0.41) NQO2BCHEIDO1KDM4EHSD17B10
SCHEMBL27411086 0.67 NQO2 (0.41) NQO2BCHEIDO1KDM4EHSD17B10
SCHEMBL8090338 0.66 GRIN1 (0.53)
SCHEMBL3635747 0.66 NQO2 (0.49) NQO2IDO1KDM4EHSD17B10ALDH1A1
SCHEMBL2552330 0.66 AAK1 (0.50) NQO2IDO1KDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2276748-A1 BICYCLIC NITROGEN CONTAINING HETEROCYCLIC COMPOUNDS FOR USE AS STEAROYL COA DESATURASE INHIBITORS Gilead Sciences, Inc. (US) 2011-01-26 EP disclosed
WO-2009126123-A1 BICYCLIC NITROGEN CONTAINING HETEROCYCLIC COMPOUNDS FOR USE AS STEAROYL COA DESATURASE INHIBITORS CV THERAPEUTICS INC. (US) 2009-10-15 WO disclosed