SCHEMBL906377

SCHEMBL906377

Cc1nc2c(CCNC(=O)OC(C)(C)C)cc(Br)cc2[nH]c1=O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.41
CACNA1H O95180 1/20 0.41
CACNA1B Q00975 1/20 0.41
CACNA1C Q13936 1/20 0.41
KDM4E B2RXH2 10/20 0.39
HSD17B10 Q99714 10/20 0.39
TSHR P16473 5/20 0.39
BCHE P06276 1/20 0.39
IDO1 P14902 2/20 0.38
ALDH1A1 P00352 7/20 0.38
CYP1A2 P05177 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HPGD P15428 4/20 0.36
GFER P55789 1/20 0.36
USP2 O75604 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL906519 0.87 CACNA1H (0.43) NQO2CACNA1HCACNA1BCACNA1CKDM4E
SCHEMBL3431673 0.78 HSD17B10 (0.41) KDM4EHSD17B10TSHRALDH1A1CYP1A2
SCHEMBL3844306 0.74 IDO1 (0.48) NQO2KDM4EHSD17B10IDO1ALDH1A1
SCHEMBL7841704 0.69 MTNR1A (0.51) NQO2KDM4EHSD17B10TSHRBCHE
SCHEMBL13400107 0.69 CA1 (0.46) NQO2KDM4EIDO1ALDH1A1NPSR1
SCHEMBL29888968 0.69 NQO2 (0.50) NQO2KDM4EHSD17B10IDO1ALDH1A1
SCHEMBL27411086 0.69 NQO2 (0.41) NQO2KDM4EHSD17B10TSHRBCHE
SCHEMBL30981863 0.69 NQO2 (0.41) NQO2KDM4EHSD17B10TSHRBCHE
SCHEMBL17942099 0.68 NPSR1 (0.50) NQO2TSHRBCHEIDO1ALDH1A1
SCHEMBL8090338 0.68 GRIN1 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2276748-A1 BICYCLIC NITROGEN CONTAINING HETEROCYCLIC COMPOUNDS FOR USE AS STEAROYL COA DESATURASE INHIBITORS Gilead Sciences, Inc. (US) 2011-01-26 EP disclosed
WO-2009126123-A1 BICYCLIC NITROGEN CONTAINING HETEROCYCLIC COMPOUNDS FOR USE AS STEAROYL COA DESATURASE INHIBITORS CV THERAPEUTICS INC. (US) 2009-10-15 WO disclosed