SCHEMBL9067778

SCHEMBL9067778

COc1ccc(-n2c(C(C)NCCN(C)C)nc3ccccc3c2=O)cc1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 4/20 0.59
ALDH1A1 P00352 4/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
LMNA P02545 1/20 0.52
PDE10A Q9Y233 4/20 0.52
RAB9A P51151 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
GAA P10253 1/20 0.48
PTGS2 P35354 1/20 0.48
TSHR P16473 1/20 0.48
KCNH2 Q12809 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
G6PD P11413 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7699242 0.90 CXCR3 (0.48) CXCR3ALDH1A1MEN1KMT2ACYP1A2
SCHEMBL7144891 0.88 CXCR3 (0.62) CXCR3PDE10A
SCHEMBL5156390 0.85 CXCR3 (0.46) CXCR3KCNH2HRH3
SCHEMBL7010507 0.83 HRH3 (0.64) ALDH1A1MEN1KMT2ACYP1A2CYP3A4
SCHEMBL452172 0.83 ALDH1A1 (0.61) CXCR3ALDH1A1MEN1KMT2ACYP1A2
SCHEMBL12672493 0.80 MAPT (0.54) CXCR3ALDH1A1MEN1KMT2ALMNA
SCHEMBL451255 0.78 ALDH1A1 (0.64) CXCR3ALDH1A1MEN1KMT2ACYP1A2
SCHEMBL12672676 0.77 PIK3CD (0.50) CXCR3LMNAPDE10AKCNH2HRH3
SCHEMBL15457233 0.76 C1R (0.45) CXCR3ALDH1A1MEN1KMT2ACYP1A2
SCHEMBL1888478 0.76 MAPT (0.52) CXCR3ALDH1A1MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216232-A1 HETEROCYCLIC COMPOUNDS AND METHODS FOR MODULATING CXCR3 FUNCTION Chemocentryx, Inc. (US) 2002-06-26 EP disclosed
WO-2001016114-A2 HETEROCYCLIC COMPOUNDS AND METHODS FOR MODULATING CXCR3 FUNCTION CHEMOCENTRYX, INC. (US) 2001-03-08 WO disclosed