SCHEMBL9068531

SCHEMBL9068531

CC(=O)SCC(CC(C)C)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)O

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 6/20 0.75
ACE P12821 2/20 0.64
MMP2 P08253 5/20 0.64
MMP9 P14780 4/20 0.64
MMP8 P22894 4/20 0.64
MMP1 P03956 2/20 0.64
ANPEP P15144 1/20 0.60
ERAP2 Q6P179 1/20 0.60
ERAP1 Q9NZ08 1/20 0.60
ALOX15 P16050 1/20 0.60
ADAM10 O14672 1/20 0.59
ADAM12 O43184 1/20 0.59
ADAMTS4 O75173 1/20 0.59
MMP3 P08254 1/20 0.59
MMP7 P09237 1/20 0.59
MMP12 P39900 1/20 0.59
MMP13 P45452 1/20 0.59
MMP14 P50281 1/20 0.59
MMP15 P51511 1/20 0.59
MMP16 P51512 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11430738 0.93 ACE (0.67) ECE1ACEALOX15
SCHEMBL7322267 0.90 ACE (0.73) ECE1ACEALOX15
SCHEMBL6172205 0.89 LTA4H (0.69) ECE1ACEALOX15
SCHEMBL6172199 0.89 LTA4H (0.69) ECE1ACEALOX15
SCHEMBL6575025 0.86 MMP2 (0.85) ECE1ACEMMP2MMP9MMP8
SCHEMBL9068557 0.86 ECE1 (1.00) ECE1ACE
SCHEMBL4795667 0.86 MMP2 (0.85) ECE1ACEMMP2MMP9MMP8
SCHEMBL6171219 0.85 MME (0.71) ECE1ACEALOX15
SCHEMBL6431194 0.85 ECE1 (0.79) ECE1ACEMMP2MMP9MMP8
SCHEMBL31036126 0.85 ECE1 (0.79) ECE1ACEMMP2MMP9MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5496805-A DIURETIC, HYPOTENSIVE E. R. SQUIBB & SONS, INC. (US) 1996-03-05 US disclosed