SCHEMBL9069237

SCHEMBL9069237

CC(=O)Br.O=C(O)C[C@H](NC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 15/20 0.60
MME P08473 1/20 0.55
ECE1 P42892 1/20 0.55
ALDH1A1 P00352 1/20 0.54
ALOX15 P16050 1/20 0.54
CTSK P43235 3/20 0.53
CTSL P07711 1/20 0.52
CTSB P07858 1/20 0.52
CTSS P25774 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL613386 0.93 CASP1 (0.67) CASP1MMEECE1
SCHEMBL554032 0.93 CASP1 (0.67) CASP1MMEECE1
SCHEMBL376886 0.93 CASP1 (0.67) CASP1MMEECE1
SCHEMBL9069236 0.88 CASP1 (0.59) CASP1MMEECE1
SCHEMBL10605640 0.88 PPARA (0.62) CASP1MMEECE1
SCHEMBL10789378 0.88 MME (0.62) CASP1MMEECE1CTSK
SCHEMBL7318257 0.88 ALDH1A1 (0.65) ALDH1A1ALOX15CTSKCTSLCTSB
SCHEMBL13007019 0.87 CASP1 (0.64) CASP1ALDH1A1ALOX15CTSKCTSL
SCHEMBL15381004 0.87 CASP1 (0.64) CASP1ALDH1A1ALOX15CTSKCTSL
SCHEMBL4405472 0.87 ALDH1A1 (0.57) CASP1ALDH1A1ALOX15CTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1504462-A Pyrimidinyl derivatives as interleukin inhibitors ������˹ҩƷ��˾ 2004-06-16 CN disclosed
CN-1118458-C Pyrimidinyl derivatives as interleukin inhibitors FERTERX PHARMACEUTICAL INC (US) 2003-08-20 CN disclosed
CN-1149292-A Pyrimidinyl derivatives as interleukin inhibitors SANOFI WINTHROP INC (US) 1997-05-07 CN disclosed
US-5585357-A Heteroaryloxymethyl ketones as interleukin-1βconverting enzyme inhibitors SANOFI WINTHROP INC. (US) 1996-12-17 US disclosed
EP-0644198-A1 Alpha-heteroaryloxymethyl ketones as interleukin-1beta converting enzyme inhibitors STERLING WINTHROP INC. (US) 1995-03-22 EP disclosed