SCHEMBL9075652

SCHEMBL9075652

C=CC[CH]c1ccncc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SNCA P37840 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.38
HDAC8 Q9BY41 1/20 0.38
JUN P05412 1/20 0.37
NFKB1 P19838 1/20 0.37
CYP19A1 P11511 2/20 0.35
CYP11B2 P19099 2/20 0.35
MAPT P10636 5/20 0.35
LMNA P02545 1/20 0.35
NPC1 O15118 4/20 0.34
RAB9A P51151 3/20 0.34
KDM4E B2RXH2 2/20 0.34
HPGD P15428 2/20 0.34
CYP1A2 P05177 2/20 0.34
MEN1 O00255 1/20 0.34
ALOX15 P16050 1/20 0.34
CASP1 P29466 1/20 0.34
HBB P68871 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8198472 0.78 JUN (0.36) SNCASMN1; SMN2JUNNFKB1CYP19A1
SCHEMBL7803558 0.77
SCHEMBL27551922 0.76 SNCA (0.35) SNCASMN1; SMN2JUNNFKB1CYP19A1
SCHEMBL288700 0.74
SCHEMBL87669 0.74 ALDH1A1 (0.52) SMN1; SMN2CYP19A1LMNAMEN1KMT2A
SCHEMBL8474249 0.73 CYP11B2 (0.50) SMN1; SMN2JUNNFKB1CYP19A1CYP11B2
SCHEMBL28222778 0.73 ALDH1A1 (0.59) SMN1; SMN2HDAC8JUNNFKB1CYP19A1
SCHEMBL14867 0.73
SCHEMBL1515220 0.72
SCHEMBL28016850 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5550233-A AUTOIMMUNE DISEASES; PREVENTION OF TRANSPLANT REJECTION MERCK & CO., INC. (US) 1996-08-27 US claimed
US-5252732-A D-heteroaryl, O-alkylheteroaryl, O-alkenylheteroaryl and O-alkynylheteroarylmacrolides having immunosuppressive activity MERCK & CO., INC. (US) 1993-10-12 US claimed
US-5550233-A AUTOIMMUNE DISEASES; PREVENTION OF TRANSPLANT REJECTION MERCK & CO., INC. (US) 1996-08-27 US disclosed
US-5349061-A O-heteroaryl, O-alkylheteroaryl, O-alkenylheteroaryl and O-alkynylheteroarylmacrolides having immunosuppressive activity MERCK & CO., INC. (US) 1994-09-20 US disclosed
US-5252732-A D-heteroaryl, O-alkylheteroaryl, O-alkenylheteroaryl and O-alkynylheteroarylmacrolides having immunosuppressive activity MERCK & CO., INC. (US) 1993-10-12 US disclosed