SCHEMBL9075694

SCHEMBL9075694

O=C(CCCNC(=O)OCc1ccccc1)NCC1CCCN1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.56
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
HDAC3 O15379 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC10 Q969S8 1/20 0.50
HDAC11 Q96DB2 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
HDAC9 Q9UKV0 1/20 0.50
HDAC5 Q9UQL6 1/20 0.50
NCOR2 Q9Y618 1/20 0.50
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
GAA P10253 1/20 0.46
TGM2 P21980 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9075691 1.00 HTT (0.56) HTTMEN1KMT2AHDAC3HDAC4
SCHEMBL4154315 0.88 ALDH1A1 (0.52) HTTMEN1KMT2AALDH1A1LMNA
SCHEMBL4741712 0.88 ALDH1A1 (0.52) HTTMEN1KMT2AALDH1A1LMNA
SCHEMBL8246719 0.88 ALDH1A1 (0.52) HTTMEN1KMT2AALDH1A1LMNA
Hydrochloric Acid SCHEMBL4741714 0.86 ALDH1A1 (0.51) HTTMEN1KMT2AALDH1A1LMNA
Hydrochloric Acid SCHEMBL4741718 0.86 ALDH1A1 (0.51) HTTMEN1KMT2AALDH1A1LMNA
SCHEMBL28351994 0.84 ALDH1A1 (0.54) HTTMEN1KMT2AALDH1A1LMNA
SCHEMBL21041192 0.84 ALDH1A1 (0.54) HTTMEN1KMT2AALDH1A1LMNA
SCHEMBL8696499 0.80 LTA4H (0.42) MEN1KMT2AALDH1A1DPP4DPP8
SCHEMBL15548368 0.78 HDAC3 (0.78) HTTHDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5583146-A Heterocyclic thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-10 US disclosed
EP-0623596-A1 N-acylpyrrolidines or N-acylpiperidines having a guanidinyl- or amidinyl-substituted side chain as thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1994-11-09 EP disclosed