SCHEMBL9076485

SCHEMBL9076485

NCc1ccc(NCC2CCCN2C(=O)C(N)Cc2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 7/20 0.58
DPP8 Q6V1X1 4/20 0.58
DPP9 Q86TI2 4/20 0.58
DPP7 Q9UHL4 4/20 0.58
FAP Q12884 2/20 0.58
F2 P00734 3/20 0.50
PRSS1 P07477 1/20 0.50
TACR1 P25103 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9076481 1.00 DPP4 (0.58) DPP4DPP8DPP9DPP7FAP
SCHEMBL9076445 0.87 DPP4 (0.55) DPP4DPP8DPP9DPP7FAP
SCHEMBL8191997 0.80 DPP4 (0.61) DPP4DPP8DPP9DPP7FAP
SCHEMBL6164069 0.80 DPP4 (0.67) DPP4DPP8DPP9DPP7FAP
SCHEMBL9076667 0.78 F2 (0.63) F2
SCHEMBL9076665 0.78 F2 (0.63) F2
SCHEMBL7102492 0.77 CYP3A4 (0.58) DPP4DPP8DPP9DPP7FAP
SCHEMBL8699172 0.76 DPP4 (0.56) DPP4DPP8DPP9DPP7FAP
SCHEMBL6164541 0.75 F2 (0.62) DPP4DPP8DPP9DPP7FAP
SCHEMBL6162266 0.75 DPP4 (0.73) DPP4DPP8DPP9DPP7FAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5583146-A Heterocyclic thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-10 US disclosed
EP-0623596-A1 N-acylpyrrolidines or N-acylpiperidines having a guanidinyl- or amidinyl-substituted side chain as thrombin inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 1994-11-09 EP disclosed