SCHEMBL907903

SCHEMBL907903

Cc1n[nH]c(=O)cc1C(C)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.40
HCAR2 Q8TDS4 2/20 0.35
HCAR3 P49019 2/20 0.35
DAO P14920 1/20 0.34
JAK1 P23458 1/20 0.34
THRA P10827 2/20 0.34
THRB P10828 2/20 0.34
PTGS2 P35354 6/20 0.33
PTGS1 P23219 2/20 0.33
ALDH1A1 P00352 1/20 0.33
AKR1B1 P15121 1/20 0.32
HSD17B10 Q99714 1/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3220976 0.69 CHEK1 (0.40) POLBDAOPTGS2PTGS1ALDH1A1
SCHEMBL4059035 0.68 ALDH1A1 (0.45) POLBPTGS2ALDH1A1AKR1B1KDM4E
SCHEMBL8404400 0.66
SCHEMBL907718 0.66 HCAR3 (0.34) POLBHCAR2HCAR3DAOJAK1
SCHEMBL909421 0.66 HCAR2 (0.46) POLBHCAR2HCAR3DAOPTGS2
SCHEMBL9696621 0.64 POLB (0.35) POLBHCAR2HCAR3ALDH1A1
SCHEMBL11458159 0.64 ALDH1A1 (0.56) POLBPTGS2ALDH1A1HSD17B10KDM4E
SCHEMBL11470412 0.64 KDM4E (0.46) PTGS2PTGS1ALDH1A1KDM4ELMNA
SCHEMBL7629389 0.63 GRM1 (0.42) PTGS2PTGS1ALDH1A1HSD17B10KDM4E
SCHEMBL27037937 0.63 HCAR2 (0.46) HCAR2DAOJAK1HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2276756-A1 HYDROXYMETHYL PYRROLIDINES AS BETA 3 ADRENERGIC RECEPTOR AGONISTS Merck Sharp & Dohme Corp. (US) 2011-01-26 EP disclosed
WO-2009124166-A1 HYDROXYMETHYL PYRROLIDINES AS BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK & CO., INC. (US) 2009-10-08 WO disclosed
WO-2009124167-A1 HYDROXYMETHYL PYRROLIDINES AS BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK & CO., INC. (US) 2009-10-08 WO disclosed