SCHEMBL9079903

SCHEMBL9079903

O=C1N(N2CCCCC2)c2ccccc2C1(Cc1ccnc(F)c1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ2 O43526 3/20 0.46
CYP3A4 P08684 2/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
ADRA1D P25100 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
KCNH2 Q12809 1/20 0.46
PDE4A P27815 5/20 0.35
PDE4B Q07343 5/20 0.35
PDE4C Q08493 5/20 0.35
PDE4D Q08499 5/20 0.35
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
THPO P40225 1/20 0.33
SCN9A Q15858 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8873348 0.90 KCNQ2 (0.44) KCNQ2CYP3A4ALOX15TSHRADRA1D
SCHEMBL8873632 0.85 CYP1A2 (0.47) KCNQ2CYP3A4ALOX15TSHRPDE4A
SCHEMBL8874782 0.83 PDE4A (0.36) CYP3A4TSHRPDE4APDE4BPDE4C
SCHEMBL8874764 0.77 KCNQ2 (0.50) KCNQ2CYP3A4ALOX15TSHRADRA1D
Water SCHEMBL9391496 0.76 KCNQ2 (0.49) KCNQ2CYP3A4ALOX15TSHRADRA1D
Water SCHEMBL9391493 0.76 KCNQ2 (0.49) KCNQ2CYP3A4ALOX15TSHRADRA1D
SCHEMBL8873879 0.74 ALDH1A1 (0.46) KCNQ2CYP3A4ALOX15TSHRPDE4A
SCHEMBL8874861 0.72 ALDH1A1 (0.37) CYP3A4TSHRKCNH2ALDH1A1CYP1A2
SCHEMBL8873140 0.71 ALDH1A1 (0.57) KCNQ2CYP3A4ALOX15TSHRPDE4A
SCHEMBL8873178 0.70 ALDH1A1 (0.46) CYP3A4TSHRALDH1A1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5519132-A ALZHEIMER*S DISEASE, NERVOUS SYSTEM DISORDERS, PROMOTE RELEASE OF ACETYLCHOLINE THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-05-21 US disclosed
WO-1994007891-A1 1-SUBSTITUTED OXINDOLES AND AZAOXINDOLES AS NOVEL COGNITION ENHANCERS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1994-04-14 WO disclosed