SCHEMBL9080475

SCHEMBL9080475

C=CCC(C#N)(CC)c1cccc(O)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.37
ALDH1A1 P00352 3/20 0.36
CYP3A4 P08684 2/20 0.36
TSHR P16473 2/20 0.34
KIF11 P52732 4/20 0.33
OPRM1 P35372 3/20 0.33
OPRD1 P41143 2/20 0.33
OPRK1 P41145 2/20 0.33
HTT P42858 1/20 0.33
AR P10275 1/20 0.32
DRD2 P14416 1/20 0.32
DRD1 P21728 1/20 0.32
DRD4 P21917 1/20 0.32
DRD5 P21918 1/20 0.32
DRD3 P35462 1/20 0.32
CA12 O43570 1/20 0.31
CA2 P00918 1/20 0.31
LMNA P02545 1/20 0.31
CA5A P35218 1/20 0.31
CA9 Q16790 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9080465 0.91 ALDH1A1 (0.38) ACHEALDH1A1CYP3A4TSHRKIF11
SCHEMBL9079288 0.88 ALDH1A1 (0.42) ACHEALDH1A1CYP3A4TSHRKIF11
SCHEMBL8031704 0.81 ALDH1A1 (0.43) ALDH1A1CYP3A4TSHROPRM1HTT
SCHEMBL8031703 0.81 ALDH1A1 (0.43) ALDH1A1CYP3A4TSHROPRM1HTT
SCHEMBL8031705 0.81 ALDH1A1 (0.43) ALDH1A1CYP3A4TSHROPRM1HTT
SCHEMBL9079258 0.80 KIF11 (0.37) ACHEALDH1A1CYP3A4KIF11AR
SCHEMBL9081259 0.78 ATM (0.45) KIF11OPRM1OPRD1OPRK1DRD2
SCHEMBL4430846 0.75 TP53 (0.39) ACHEALDH1A1CYP3A4TSHRKIF11
SCHEMBL15242489 0.73 MAPT (0.46) ACHEALDH1A1CYP3A4TSHRKIF11
SCHEMBL9080223 0.73 PRKCQ (0.44) ACHEALDH1A1CYP3A4TSHRKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5519022-A α, α dialkylbenzyl derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1996-05-21 US disclosed
US-5288742-A Lipoxygenase inhibitor IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-02-22 US disclosed
EP-0505122-A1 Alpha, alpha-dialkylbenzyl derivatives ZENECA LIMITED (GB) 1992-09-23 EP disclosed