SCHEMBL9079258

SCHEMBL9079258

C=CCC(C#N)(CC)c1cccc(OC)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.37
PDE4A P27815 3/20 0.37
PDE4B Q07343 3/20 0.37
PDE4C Q08493 3/20 0.37
PDE4D Q08499 3/20 0.37
PGR P06401 1/20 0.36
AR P10275 1/20 0.36
CASP1 P29466 1/20 0.36
HSD17B10 Q99714 1/20 0.36
NPC1 O15118 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALDH1A1 P00352 3/20 0.35
ALOX12 P18054 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
ACHE P22303 1/20 0.34
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
NFE2L2 Q16236 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7673680 0.93 KIF11 (0.40) KIF11PDE4APDE4BPDE4CPDE4D
SCHEMBL9079230 0.88 KIF11 (0.42) KIF11PDE4APDE4BPDE4CPDE4D
SCHEMBL9080475 0.80 ACHE (0.37) KIF11ARHSD17B10SMN1; SMN2ALDH1A1
SCHEMBL9080579 0.80 MAOB (0.43) KIF11USP2KMT2A
SCHEMBL8031705 0.79 ALDH1A1 (0.43) SMN1; SMN2ALDH1A1CYP3A4KMT2A
SCHEMBL8031703 0.79 ALDH1A1 (0.43) SMN1; SMN2ALDH1A1CYP3A4KMT2A
SCHEMBL8031704 0.79 ALDH1A1 (0.43) SMN1; SMN2ALDH1A1CYP3A4KMT2A
SCHEMBL4874767 0.75 CASP1 (0.44) KIF11PDE4APDE4BPDE4CPDE4D
SCHEMBL9080527 0.75 PRKCQ (0.43) KIF11PDE4APDE4BPDE4CPDE4D
SCHEMBL11259641 0.75 FFAR1 (0.41) PDE4BHSD17B10MAPK1ALDH1A1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5519022-A α, α dialkylbenzyl derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1996-05-21 US disclosed
US-5288742-A Lipoxygenase inhibitor IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-02-22 US disclosed
EP-0505122-A1 Alpha, alpha-dialkylbenzyl derivatives ZENECA LIMITED (GB) 1992-09-23 EP disclosed