SCHEMBL9084136

SCHEMBL9084136

CC(=O)Oc1cc(C(F)(F)F)ccc1C(=O)NCCO[N+](=O)[O-]

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
CYP2C19 P33261 2/20 0.54
HSD17B10 Q99714 2/20 0.54
HPGD P15428 2/20 0.54
KDM4E B2RXH2 1/20 0.54
USP2 O75604 1/20 0.54
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
PTGS2 P35354 2/20 0.42
MAPT P10636 5/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CYP2C9 P11712 1/20 0.41
ALOX15 P16050 1/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
LMNA P02545 3/20 0.41
POLB P06746 1/20 0.41
MCHR1 Q99705 2/20 0.39
THRB P10828 1/20 0.39
TLR2 O60603 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9085960 0.92 ALDH1A1 (0.50) ALDH1A1CYP2C19HSD17B10HPGDKDM4E
SCHEMBL4421848 0.83 KMT2A (0.45) CYP2C19HSD17B10HPGDNPC1RAB9A
SCHEMBL9083520 0.82 TP53 (0.47) ALDH1A1CYP2C19HSD17B10HPGDKDM4E
SCHEMBL9085187 0.82 PTGS2 (0.41) ALDH1A1CYP2C19HSD17B10HPGDKDM4E
SCHEMBL5943436 0.81 ALDH1A1 (0.60) ALDH1A1CYP2C19HSD17B10HPGDKDM4E
SCHEMBL9545778 0.80 PTGS2 (0.62) ALDH1A1CYP2C19HSD17B10HPGDKDM4E
SCHEMBL13142986 0.79 ALDH1A1 (0.57) ALDH1A1CYP2C19HSD17B10HPGDKDM4E
SCHEMBL9082978 0.79 PTGS2 (0.49) ALDH1A1CYP2C19HSD17B10HPGDKDM4E
SCHEMBL16190215 0.77 ALDH1A1 (0.53) ALDH1A1CYP2C19HSD17B10HPGDKDM4E
SCHEMBL9082797 0.76 MEN1 (0.50) CYP2C19HSD17B10NPC1PTGS2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5589490-A BENZAMIDE DERIVATIVES WITH NITROXY ALKYL GROUPS ITALFARMACO S.P.A. (IT) 1996-12-31 US disclosed
EP-0540544-B1 BENZOIC ACID SUBSTITUTED DERIVATIVES HAVING CARDIOVASCULAR ACTIVITY ITALFARMACO SPA (IT) 1995-02-15 EP disclosed
US-5366992-A IN MIXTURE WITH AN EXCIPIENT ITALFARMACO S.P.A. (IT) 1994-11-22 US disclosed
WO-1992001668-A1 BENZOIC ACID SUBSTITUTED DERIVATIVES HAVING CARDIOVASCULAR ACTIVITY ITALFARMACO S.P.A. (IT) 1992-02-06 WO disclosed