SCHEMBL9085501

SCHEMBL9085501

C=CCC(C)(C)CNc1cc(Cl)ncn1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.35
HRH4 Q9H3N8 3/20 0.35
HRH3 Q9Y5N1 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
FGFR4 P22455 1/20 0.32
EGFR P00533 1/20 0.31
MKNK1 Q9BUB5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9085595 0.79 ESR1 (0.38)
SCHEMBL15356370 0.79 HRH4 (0.51) NPC1HRH4HRH3MEN1KMT2A
SCHEMBL9277137 0.78 CLK4 (0.35)
SCHEMBL6696015 0.76 NPC1 (0.40) NPC1HRH4HRH3MEN1KMT2A
SCHEMBL3814997 0.76 ALDH1A1 (0.42) NPC1MEN1KMT2AMKNK1
SCHEMBL9084848 0.74 CDC7 (0.38)
SCHEMBL602892 0.73 MEN1 (0.41) NPC1HRH4HRH3MEN1KMT2A
SCHEMBL374260 0.70 EGFR (0.53) NPC1MEN1KMT2AFGFR4EGFR
SCHEMBL18131074 0.70 MEN1 (0.49) NPC1MEN1KMT2AFGFR4EGFR
SCHEMBL28158644 0.67 DNM2 (0.45) NPC1HRH4MEN1KMT2AEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5550240-A Piperazinyl-bis(alkylamino)pyrimidine derivatives and process for preparing same RICHTER GEDEON VEGYESZETI GYAR RT. (HU) 1996-08-27 US disclosed
EP-0644882-A1 NOVEL PIPERZINYL-BIS(ALKYLAMINO)PYRIMIDINE DERIVATIVES AND PROCESS FOR PREPARING SAME RICHTER GEDEON VEGYESZETI GYAR R.T. (HU) 1995-03-29 EP disclosed
WO-1993025539-A1 NOVEL PIPERZINYL-BIS(ALKYLAMINO)PYRIMIDINE DERIVATIVES AND PROCESS FOR PREPARING SAME Richter Gedeon Vegyészeti Gyár Rt. (HU) 1993-12-23 WO disclosed