SCHEMBL9092014

SCHEMBL9092014

CC(=O)OCc1cc(-c2ccc3c(c2)C=CC(C)(C)O3)ccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
COXFA4 O00483 1/20 0.44
HIF1A Q16665 9/20 0.41
EPAS1 Q99814 9/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
CYP3A4 P08684 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
PTPN1 P18031 1/20 0.39
TLR3 O15455 1/20 0.39
EP300 Q09472 4/20 0.38
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
XDH P47989 1/20 0.37
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
TP53 P04637 1/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9092543 0.86 HIF1A (0.44) COXFA4HIF1AEPAS1ALDH1A1HPGD
Acetic Acid SCHEMBL9092012 0.85 HIF1A (0.42) COXFA4HIF1AEPAS1ALDH1A1HPGD
SCHEMBL9092249 0.82 HIF1A (0.46) HIF1AEPAS1ALDH1A1HPGDCYP3A4
SCHEMBL9091985 0.80 HIF1A (0.45) HIF1AEPAS1ALDH1A1HPGDEP300
SCHEMBL9090422 0.80 HIF1A (0.45) HIF1AEPAS1ALDH1A1HPGDEP300
SCHEMBL27665986 0.78 COXFA4 (0.57) COXFA4HIF1AEPAS1ALDH1A1HPGD
SCHEMBL9092974 0.75 HIF1A (0.46) HIF1AEPAS1ALDH1A1HPGDCYP3A4
SCHEMBL12580741 0.74 ALDH1A1 (0.43) COXFA4HIF1AEPAS1ALDH1A1HPGD
SCHEMBL12095636 0.73 HSD17B10 (0.45) HSD17B10
SCHEMBL3307991 0.71 PKM (0.45) ALDH1A1KDM4ECA12CA1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5574049-A POTASSIUM CHANNEL OPENERS, BRONCHODILATORS, ANTIASTHMA SANDOZ LTD. (CH) 1996-11-12 US disclosed
EP-0623129-A1 2,2-DIALKYL- AND 2,2-DIALKYL-3,4-DIHYDRO-3-HYDROXY-2H-1-BENZOPYR ANS, THEIR USE AS PHARMACEUTICALS Novartis AG (CH) 1994-11-09 EP disclosed
WO-1994012493-A1 2,2-DIALKYL- AND 2,2-DIALKYL-3,4-DIHYDRO-3-HYDROXY-2H-1-BENZOPYR ANS, THEIR USE AS PHARMACEUTICALS SANDOZ, LTD. (CH) 1994-06-09 WO disclosed