SCHEMBL9103038

SCHEMBL9103038

CNC(=O)NCc1ccccc1-c1ccc(CN2C(=O)[C@H](NC(=O)CC(C)(C)NCc3ccco3)CSc3cc(OC)ccc32)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 4/20 0.48
TP53 P04637 3/20 0.36
AGTR1 P30556 1/20 0.35
POLB P06746 4/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
TDP1 Q9NUW8 2/20 0.35
APEX1 P27695 1/20 0.35
RECQL P46063 1/20 0.35
BLM P54132 1/20 0.35
XIAP P98170 2/20 0.35
ALDH1A1 P00352 5/20 0.34
MAPT P10636 4/20 0.33
HSD17B10 Q99714 3/20 0.33
KDM4E B2RXH2 3/20 0.33
HPGD P15428 2/20 0.33
ALOX15 P16050 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
ESR1 P03372 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9103333 0.95 GHSR (0.49) GHSRTP53AGTR1POLBMEN1
SCHEMBL9101352 0.94 GHSR (0.49) GHSRTP53AGTR1POLBMEN1
SCHEMBL9102792 0.93 GHSR (0.42) GHSRTP53AGTR1POLBMEN1
SCHEMBL9109295 0.92 GHSR (0.49) GHSRTP53AGTR1POLBKMT2A
SCHEMBL9105564 0.91 GHSR (0.54) GHSRTP53AGTR1POLBKMT2A
SCHEMBL9102858 0.91 GHSR (0.49) GHSRAGTR1POLBXIAPALDH1A1
SCHEMBL9102835 0.91 GHSR (0.48) GHSRTP53AGTR1POLBKMT2A
SCHEMBL9105585 0.89 GHSR (0.58) GHSRAGTR1XIAP
SCHEMBL7794630 0.89 GHSR (0.49) GHSRAGTR1XIAP
SCHEMBL7791658 0.89 GHSR (0.56) GHSRAGTR1XIAPMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5430144-A E.g, N-(1-((2'-((methoxycarbonyl)amino)(1,1'-biphenyl)-4-yl) methyl)-2,3,4,5-tetrahydro-2-oxo-1H-1-benzazepin-3-yl)-3 ((fur-2-yl)methyl)amino-3-methylbutanamide MERCK & CO., INC. (US) 1995-07-04 US disclosed