SCHEMBL9103685

SCHEMBL9103685

CCC(C=O)N(CCc1c[nH]c2ccccc12)C(=O)CC1C(=O)N(C(Cl)Cc2ccc(Cl)cc2)CC(=O)N1CCOC

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 1/20 0.36
CCND1 P24385 1/20 0.36
PIM1 P11309 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
HPGD P15428 2/20 0.34
TACR1 P25103 2/20 0.33
CCKBR P32239 1/20 0.33
MC4R P32245 2/20 0.32
MC3R P41968 2/20 0.32
MEN1 O00255 2/20 0.32
RAB9A P51151 2/20 0.32
KMT2A Q03164 2/20 0.32
MAPT P10636 2/20 0.32
DRD2 P14416 2/20 0.32
DRD4 P21917 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9280399 0.91 MAPT (0.37) CDK4CCND1PIM1CYP3A4CYP2D6
SCHEMBL9105301 0.89 TACR2 (0.42) CDK4CCND1PIM1CYP3A4CYP2D6
SCHEMBL9107408 0.88 LMNA (0.32) MEN1KMT2AMAPTALDH1A1LMNA
SCHEMBL3700997 0.86 APAF1 (0.38) CDK4CCND1PIM1CYP3A4CYP2D6
SCHEMBL3691829 0.81 HPGD (0.39) CDK4CCND1PIM1CYP3A4CYP2D6
SCHEMBL3698794 0.81 SMN1; SMN2 (0.42) CYP3A4CYP2D6CYP2C9CYP2C19HPGD
SCHEMBL9104168 0.80 GPBAR1 (0.32) KMT2A
SCHEMBL9279133 0.80 MAPT (0.39) CDK4CCND1PIM1CYP3A4CYP2D6
SCHEMBL3702676 0.80 DRD3 (0.37) CDK4CCND1PIM1CYP3A4CYP2D6
SCHEMBL3775360 0.79 APAF1 (0.40) CDK4CCND1PIM1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2460798-A2 APAF-1 INHIBITOR COMPOUNDS Laboratorios SALVAT, S.A. (ES) 2012-06-06 EP disclosed