SCHEMBL9107536

SCHEMBL9107536

O=C(O)C1CCc2ccccc2NC1=O

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.47
MAPK13 O15264 1/20 0.47
MAPK12 P53778 1/20 0.47
MAPK11 Q15759 1/20 0.47
MAPK14 Q16539 1/20 0.47
PYGL P06737 5/20 0.47
PYGM P11217 5/20 0.47
ALDH1A1 P00352 1/20 0.46
DDB1 Q16531 1/20 0.46
CRBN Q96SW2 1/20 0.46
MAPT P10636 2/20 0.45
RIPK1 Q13546 5/20 0.44
GAA P10253 1/20 0.42
PTK2B Q14289 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methane SCHEMBL9049828 0.98 PYGL (0.46) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL4826771 0.86 PTK2B (0.47) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL30960380 0.83 MAPT (0.53) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL219216 0.83 MAPT (0.53) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL4335722 0.77 GLA (0.47) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL4232147 0.77 PYGL (0.66) PYGLPYGMDDB1CRBNRIPK1
SCHEMBL4216634 0.77 PYGL (0.66) PYGLPYGMDDB1CRBNRIPK1
SCHEMBL1976547 0.77 PYGL (0.66) PYGLPYGMDDB1CRBNRIPK1
SCHEMBL4623734 0.76 SIRT1 (0.46) ALDH1A1
SCHEMBL12598688 0.75 NPC1 (0.52) NPC1MAPK13MAPK12MAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0382687-B1 Benzofused-N-containing heterocycle derivatives BOEHRINGER INGELHEIM ITALIA (IT) 1995-12-27 EP disclosed
WO-1995004534-A1 ENDOTHELIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1995-02-16 WO disclosed
EP-0382687-A2 Benzofused-N-containing heterocycle derivatives BOEHRINGER INGELHEIM ITALIA S.p.A. (IT) 1990-08-16 EP disclosed