SCHEMBL9113437

SCHEMBL9113437

CC(C)NC(=O)OC(C)[C@H]1CC[C@H]2[C@@H]3CCN4C(C)C(=O)CC[C@]4(C)[C@H]3CC[C@]12C

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 4/20 0.36
GPBAR1 Q8TDU6 1/20 0.35
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
CYP17A1 P05093 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9113840 0.92 GPBAR1 (0.36) SRD5A2GPBAR1FNTAFNTBCYP17A1
SCHEMBL9113792 0.89 GPBAR1 (0.36) SRD5A2GPBAR1
SCHEMBL8926995 0.86 SRD5A2 (0.33) SRD5A2
SCHEMBL8063840 0.83 GPBAR1 (0.37) SRD5A2GPBAR1FNTAFNTB
SCHEMBL8497746 0.81 GPBAR1 (0.36) SRD5A2GPBAR1FNTAFNTBCYP17A1
SCHEMBL8931575 0.80 FNTA (0.36) SRD5A2GPBAR1FNTAFNTB
SCHEMBL9114171 0.79 FAAH (0.38) SRD5A2GPBAR1FNTAFNTB
SCHEMBL7745521 0.79 RORC (0.36) SRD5A2GPBAR1FNTAFNTB
SCHEMBL8063891 0.78 SRD5A2 (0.36) SRD5A2
SCHEMBL8722384 0.78 FNTA (0.35) SRD5A2GPBAR1FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0649306-A4 ESTER DERIVATIVES OF 4-AZA-STEROIDS. MERCK & CO INC (US) 1995-08-23 EP claimed
EP-0649306-A1 ESTER DERIVATIVES OF 4-AZA-STEROIDS MERCK & CO. INC. (US) 1995-04-26 EP claimed
EP-0649306-A4 ESTER DERIVATIVES OF 4-AZA-STEROIDS. MERCK & CO INC (US) 1995-08-23 EP disclosed
EP-0649306-A1 ESTER DERIVATIVES OF 4-AZA-STEROIDS MERCK & CO. INC. (US) 1995-04-26 EP disclosed