SCHEMBL9114473

SCHEMBL9114473

O=C1OC(=O)C2=C1c1cccc3cccc2c13

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 5/20 0.74
ALDH1A1 P00352 6/20 0.58
MCL1 Q07820 2/20 0.58
CES2 O00748 1/20 0.58
BCHE P06276 1/20 0.58
CES1 P23141 1/20 0.58
PARP1 P09874 1/20 0.52
HSD17B10 Q99714 5/20 0.50
MAPK1 P28482 3/20 0.50
PABPC1 P11940 2/20 0.50
CASP1 P29466 2/20 0.50
CASP7 P55210 2/20 0.50
TSHR P16473 2/20 0.50
ATM Q13315 2/20 0.50
CYP3A4 P08684 1/20 0.50
DNMT1 P26358 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
ERCC1 P07992 1/20 0.48
FEN1 P39748 1/20 0.48
ERCC4 Q92889 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
1,8-Naphthalic Anhydride SCHEMBL30415 0.85 TYMS (1.00) TYMSALDH1A1MCL1CES2BCHE
1,8-Naphthalic Anhydride SCHEMBL29351054 0.85 TYMS (1.00) TYMSALDH1A1MCL1CES2BCHE
1,8-Naphthalic Anhydride SCHEMBL11692800 0.83 TYMS (0.95) TYMSALDH1A1MCL1CES2BCHE
1,8-Naphthalic Anhydride SCHEMBL6929962 0.83 TYMS (0.95) TYMSALDH1A1MCL1CES2BCHE
1,8-Naphthalic Anhydride SCHEMBL10012400 0.81 TYMS (0.91) TYMSALDH1A1MCL1CES2BCHE
SCHEMBL9264368 0.78 TYMS (0.47) TYMSALDH1A1MCL1CES2BCHE
1,8-Naphthalic Anhydride SCHEMBL21046340 0.77 TYMS (0.83) TYMSALDH1A1MCL1CES2BCHE
1,8-Naphthalic Anhydride SCHEMBL29143033 0.77 TYMS (0.83) TYMSALDH1A1MCL1CES2BCHE
SCHEMBL15119577 0.77 TYMS (0.75) TYMSALDH1A1MCL1CES2BCHE
SCHEMBL18845631 0.74 ALDH1A1 (0.62) TYMSALDH1A1MCL1CES2BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0683768-A1 UNSYMMETRICAL BIS-IMIDES AS ANTICANCER AGENTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-11-29 EP disclosed
WO-1995008539-A1 IMPROVED METHODS FOR PREPARING BIS-IMIDE COMPOUNDS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-03-30 WO disclosed
US-5359070-A ANTITUMOR AGENTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1994-10-25 US disclosed
WO-1994018171-A1 UNSYMMETRICAL BIS-IMIDES AS ANTICANCER AGENTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1994-08-18 WO disclosed