SCHEMBL9264368

SCHEMBL9264368

O=Cc1ccc2cccc3c2c1C1=C3C(=O)OC1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 5/20 0.47
ALDH1A1 P00352 4/20 0.37
CES1 P23141 2/20 0.37
MCL1 Q07820 2/20 0.37
CES2 O00748 1/20 0.37
BCHE P06276 1/20 0.37
POLB P06746 3/20 0.37
PTPN1 P18031 2/20 0.37
PARP1 P09874 1/20 0.34
KDM4E B2RXH2 3/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
CYP3A4 P08684 1/20 0.33
PABPC1 P11940 1/20 0.33
DNMT1 P26358 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9114473 0.78 TYMS (0.74) TYMSALDH1A1CES1MCL1CES2
SCHEMBL28471709 0.76 ALDH1A1 (0.50) TYMSALDH1A1CES1MCL1CES2
SCHEMBL548271 0.75 PARP1 (0.37) TYMSALDH1A1CES1MCL1CES2
SCHEMBL9390822 0.70 HSD17B10 (0.42) ALDH1A1CES1MCL1CES2BCHE
SCHEMBL10432889 0.70 TDP1 (0.46) TYMSALDH1A1KDM4EHPGDCYP1A2
SCHEMBL10490132 0.68 ALDH1A1 (0.48) TYMSALDH1A1CES1MCL1CES2
SCHEMBL4960210 0.68 TYMS (0.62) TYMSALDH1A1CES1MCL1CES2
SCHEMBL546727 0.68 HSD17B10 (0.40) ALDH1A1CES1MCL1CES2BCHE
1,8-Naphthalic Anhydride SCHEMBL30415 0.66 TYMS (1.00) TYMSALDH1A1CES1MCL1CES2
SCHEMBL4944634 0.66 THRB (0.52) ALDH1A1CES1MCL1CES2BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0683768-A1 UNSYMMETRICAL BIS-IMIDES AS ANTICANCER AGENTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-11-29 EP disclosed
US-5359070-A ANTITUMOR AGENTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1994-10-25 US disclosed